Ufiprazole

Ufiprazole

SCHEMBL662986

COc1ccc2[nH]c(SCc3ncc(C)c(OC)c3C)nc2c1

nearest known ligand 0.84

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 3/20 0.84
CYP2C9 P11712 12/20 0.52
CYP2C19 P33261 11/20 0.52
CYP1A2 P05177 10/20 0.52
CYP3A4 P08684 10/20 0.52
KMT2A Q03164 4/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
WDR5 P61964 2/20 0.52
HTT P42858 2/20 0.52
KDM4E B2RXH2 1/20 0.52
DDAH1 O94760 1/20 0.52
ABCB11 O95342 1/20 0.52
ALDH1A1 P00352 1/20 0.52
ATP1A1 P05023 1/20 0.52
ATP1B1 P05026 1/20 0.52
CHRM2 P08172 1/20 0.52
ABCB1 P08183 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
MAPT P10636 1/20 0.52
CHRM1 P11229 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ufiprazole SCHEMBL29455226 1.00 BRS3 (0.84) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL7929368 0.99 BRS3 (0.82) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL7950477 0.99 BRS3 (0.82) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL31529606 0.99 BRS3 (0.82) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL3180530 0.95 BRS3 (0.76) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL3170203 0.94 BRS3 (0.74) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL12873280 0.93 BRS3 (0.73) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL3186458 0.92 BRS3 (0.71) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL1816535 0.91 BRS3 (1.00) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL29693729 0.91 BRS3 (1.00) BRS3CYP2C9CYP2C19CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 725 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118271289-A Preparation method of esomeprazole sodium 苏州东瑞制药有限公司 2024-07-02 CN claimed
CN-114478481-B Preparation method of omeprazole 扬州大学 2024-04-02 CN claimed
CN-115305243-B Baeyer-Villiger monooxygenase mutant and application thereof 江南大学 2023-06-02 CN claimed
CN-115044566-B Cyclohexanone monooxygenase mutant and application thereof 江南大学 2023-05-02 CN claimed
CN-115305243-A Baeyer-Villiger monooxygenase mutant and application thereof 江南大学 2022-11-08 CN claimed
CN-112255352-B Method for detecting related substances of esomeprazole sodium for injection 海南卫康制药(潜山)有限公司 2022-10-14 CN claimed
CN-115044566-A Cyclohexanone monooxygenase mutant and application thereof 江南大学 2022-09-13 CN claimed
US-20220267742-A1 NADPH-REGENERATION SYSTEM BASED ON MONOMERIC ISOCITRATE DEHYDROGENASE AND USE THEREOF INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2022-08-25 US claimed
US-11236309-B2 Recombinant vector and method for producing reconstituted cytochrome P450 oxygenase-reductase fusion protein using the same INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2022-02-01 US claimed
US-20220016099-A1 BENZIMIDAZOLE OR BENZOXAZOLE DERIVATIVES FOR PREVENTING AND TREATING CENTRAL NERVOUS SYSTEM DISEASE, DIABETES, AND COMPLICATIONS THEREOF TRINUERO (KR) 2022-01-20 US claimed
EP-0931076-A1 METHOD OF OMEPRAZOLE PREPARATION Slovakofarma, A.S. (SK) 1999-07-28 EP claimed
WO-1999025711-A1 NEW PROCESS ASTRA AKTIEBOLAG (SE) 1999-05-27 WO claimed
WO-1998054171-A1 NOVEL FORM OF S-OMEPRAZOLE ASTRA AKTIEBOLAG (SE) 1998-12-03 WO claimed
WO-1998009962-A1 METHOD OF OMEPRAZOLE PREPARATION SLOVAKOFARMA, A.S. (SK) 1998-03-12 WO claimed
EP-0533752-B1 IMPROVED METHOD FOR SYNTHESIS ASTRA AB (SE) 1998-01-28 EP claimed
US-5578732-A MONO-OXIDATION OF SULFUR ATOM BY HYDROGEN PEROXIDE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-11-26 US claimed
US-5386032-A Method of synthesis of 5-methoxy-2-[(4-methoxy-3,5-dimethyl-2-pyridinyl)-methyl]sulfinyl-1H-benzimidazole (omeprazole) AKTIEBOLAGET ASTRA (SE) 1995-01-31 US claimed
EP-0533752-A1 IMPROVED METHOD FOR SYNTHESIS Astra Aktiebolag (SE) 1993-03-31 EP claimed
EP-0484265-A1 A process for the preparation of omeprazol CENTRO GENESIS PARA LA INVESTIGACION, S.L. (ES) 1992-05-06 EP claimed
WO-1991018895-A1 IMPROVED METHOD FOR SYNTHESIS AKTIEBOLAGET ASTRA (SE) 1991-12-12 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220016099-A1 BENZIMIDAZOLE OR BENZOXAZOLE DERIVATIVES FOR PREVENTING AND TREATING CENTRAL NERVOUS SYSTEM DISEASE, DIABETES, AND COMPLICATIONS THEREOF KEAP1, SLC5A1, GCLC BRS3 2502/4885CYP2C9 1053/4885CYP2C19 1226/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.