SCHEMBL10735166

SCHEMBL10735166

O=C(O)/C=C/C(=O)c1cccnc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 5/20 0.68
CYP1A2 P05177 5/20 0.68
CYP1B1 Q16678 5/20 0.68
CYP3A4 P08684 3/20 0.68
CYP2D6 P10635 3/20 0.68
FTO Q9C0B1 1/20 0.62
ALDH1A1 P00352 4/20 0.60
APP P05067 2/20 0.60
GAA P10253 1/20 0.60
HCAR3 P49019 1/20 0.60
HCAR2 Q8TDS4 1/20 0.60
GPR52 Q9Y2T5 1/20 0.59
MAPT P10636 5/20 0.58
KMT2A Q03164 2/20 0.56
LMNA P02545 1/20 0.56
HPGD P15428 1/20 0.56
GSK3B P49841 1/20 0.55
KDM4E B2RXH2 1/20 0.54
MEN1 O00255 1/20 0.54
NPC1 O15118 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10735172 1.00 CYP1A1 (0.68) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL1322029 0.85 CYP1A1 (0.82) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL1322027 0.85 CYP1A1 (0.82) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
Niacinamide SCHEMBL27641063 0.84 F7 (0.79) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
Niacinamide SCHEMBL19876218 0.84 F7 (0.79) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
Niacinamide SCHEMBL27698255 0.84 F7 (0.79) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
Niacinamide SCHEMBL29204086 0.84 F7 (0.79) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL10036802 0.83 CYP1A1 (0.65) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL27497512 0.83 CYP1A1 (0.65) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6
SCHEMBL10001058 0.81 CYP1A1 (0.63) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4710508-A ANALGESICS WARNER-LAMBERT COMPANY (US) 1987-12-01 US disclosed