SCHEMBL10736716

SCHEMBL10736716

Nc1ccnc(SCC#CCN2C(=O)c3ccccc3C2=O)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.50
ALDH1A1 P00352 6/20 0.38
TSHR P16473 2/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
GAA P10253 2/20 0.36
POLB P06746 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
PKM P14618 2/20 0.36
ALOX5AP P20292 2/20 0.36
FEN1 P39748 2/20 0.36
HSD17B10 Q99714 2/20 0.36
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10682225 0.80 MAPK1 (0.55) MAPK1ALDH1A1TSHRRAB9AL3MBTL1
SCHEMBL10674136 0.78 CYP1A2 (0.55) MAPK1ALDH1A1TSHRRAB9AGAA
SCHEMBL10679952 0.77 MAPK1 (0.51) MAPK1ALDH1A1TSHRRAB9AGAA
SCHEMBL10741890 0.73 MAPK1 (0.38) MAPK1ALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL11282464 0.72 MAPK1 (0.37) MAPK1ALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL9698514 0.67 ALDH1A1 (0.49) MAPK1ALDH1A1TSHRHTTGAA
SCHEMBL9084403 0.66 MAPK1 (0.71) MAPK1ALDH1A1TSHRRAB9AL3MBTL1
SCHEMBL10676066 0.65 GAA (0.46) MAPK1ALDH1A1TSHRRAB9AL3MBTL1
SCHEMBL1862779 0.64 ALDH1A1 (0.49) MAPK1ALDH1A1TSHRHTTRAB9A
SCHEMBL6357561 0.64 DRD3 (0.51) MAPK1ALDH1A1TSHRHTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4657908-A Carbonyl derivatives ICI AMERICAS, INC. (US) 1987-04-14 US disclosed
EP-0059597-B1 GUANIDINO-SUBSTITUTED HETEROCYCLIC DERIVATIVES HAVING HISTAMINE H-2 ANTAGONIST ACTIVITY IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-04-23 EP disclosed
US-4496571-A GUANIDINE DERIVATIVE ICI AMERICAS INC. (US) 1985-01-29 US disclosed
EP-0059597-A2 Guanidino-substituted heterocyclic derivatives having histamine H-2 antagonist activity IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-09-08 EP disclosed