SCHEMBL1074065

SCHEMBL1074065

COCCCc1cc(C(=O)NC2CC2)ccc1C

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 10/20 0.51
MAPK11 Q15759 3/20 0.47
CYP2C9 P11712 2/20 0.47
HSPB1 P04792 1/20 0.47
DRD4 P21917 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
KMT2A Q03164 1/20 0.44
RIPK2 O43353 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
SMYD3 Q9H7B4 1/20 0.44
TP53 P04637 1/20 0.44
TSHR P16473 1/20 0.44
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8238436 0.84 MAPK14 (0.52) MAPK14CYP2C9KMT2ASMYD3GAA
SCHEMBL1518227 0.80 MAPK14 (0.44) MAPK14CYP2C9KMT2ASMN1; SMN2ALDH1A1
SCHEMBL1070915 0.77 MEN1 (0.48) MAPK14CYP2C9KMT2ASMN1; SMN2SMYD3
SCHEMBL10282601 0.76 GLA (0.64) MAPK14MAPK11CYP2C9HSPB1NPC1
SCHEMBL661051 0.75 BRD4 (0.47) MAPK14CYP2C9NPC1KMT2ASMN1; SMN2
SCHEMBL89015 0.74 CNR2 (0.55) MAPK14CYP2C9NPC1RAB9AKMT2A
SCHEMBL90498 0.74 CNR2 (0.61) MAPK14CYP2C9KMT2ATP53
SCHEMBL27973124 0.74 ALDH1A1 (0.41) RAB9AKMT2ATSHRALDH1A1GAA
SCHEMBL2087745 0.73 LRRK2 (0.49) MAPK14RAB9AKMT2ARIPK2SMN1; SMN2
SCHEMBL27973149 0.73 MEN1 (0.36) MAPK14RAB9AKMT2ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274295-A1 3, 4 - SUBSTITUTED PIPERIDINE DERIVATIVES AS RENIN INHIBITORS Merck Frosst Canada Ltd. (CA) 2011-01-19 EP disclosed