SCHEMBL10740705

SCHEMBL10740705

O=C1CCCCC1C(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.64
MAPK1 P28482 1/20 0.60
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
BACE1 P56817 1/20 0.44
KDM2B Q8NHM5 2/20 0.44
HSD11B1 P28845 1/20 0.44
MGLL Q99685 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MEN1 O00255 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
KMT2A Q03164 1/20 0.43
DGAT1 O75907 1/20 0.42
HPD P32754 1/20 0.42
LMNA P02545 1/20 0.41
SRD5A2 P31213 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10885557 0.87 MCL1 (0.82) MCL1MAPK1ALDH1A1HPGDKMT2A
SCHEMBL1720192 0.84 MAPK1 (0.64) MCL1MAPK1ALDH1A1MEN1HPGD
SCHEMBL1720821 0.82 MCL1 (0.70) MCL1MAPK1CES2CES1HSD11B1
SCHEMBL8131947 0.81 MCL1 (0.68) MCL1MAPK1HSD11B1ALDH1A1
SCHEMBL7922437 0.79 MCL1 (0.70) MCL1MAPK1ALDH1A1TSHRLMNA
SCHEMBL27314925 0.79 MCL1 (0.70) MCL1MAPK1MGLLALDH1A1HPGD
SCHEMBL8144387 0.79 MCL1 (0.70) MCL1MAPK1CES2CES1MGLL
SCHEMBL1720195 0.79 MCL1 (0.70) MCL1MAPK1CES2CES1ALDH1A1
SCHEMBL600072 0.78 MCL1 (1.00) MCL1MAPK1ALDH1A1LMNA
SCHEMBL1855141 0.78 HSD11B1 (0.60) CES2CES1KDM2BHSD11B1MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4652559-A ANALGESIC, ANTIDEPRESSANT THE UPJOHN COMPANY (US) 1987-03-24 US disclosed
EP-0085811-B1 2-(PHENYLMETHYLENE)CYCLOALKYLAMINES THE UPJOHN COMPANY (US) 1986-05-07 EP disclosed
US-4540690-A ANALGESICS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1985-09-10 US disclosed
EP-0085811-A1 2-(Phenylmethylene)cycloalkylamines THE UPJOHN COMPANY (US) 1983-08-17 EP disclosed