SCHEMBL10748545

SCHEMBL10748545

CCN(CCO)CCNc1nnc(-c2ccccc2)cc1C

nearest known ligand 0.84

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.52
LMNA P02545 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CHRM1 P11229 1/20 0.50
CNR1 P21554 1/20 0.50
HTR2B P41595 1/20 0.50
KCNH2 Q12809 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
TP53 P04637 1/20 0.45
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1752852 0.85 ACHE (0.56) ACHELMNACYP3A4CYP1A2CYP2D6
SCHEMBL1752885 0.83 ACHE (0.62) ACHELMNACYP3A4CYP1A2CYP2D6
SCHEMBL1752857 0.80 ACHE (0.68) ACHELMNACYP3A4CYP1A2CYP2D6
SCHEMBL1752803 0.80 ACHE (0.58) ACHELMNACYP3A4CYP1A2CYP2D6
SCHEMBL1752884 0.79 ACHE (0.57) ACHELMNACYP3A4CYP1A2CYP2D6
SCHEMBL1753027 0.77 ACHE (0.48) ACHELMNACYP3A4CYP1A2CYP2D6
SCHEMBL2760423 0.76 ACHE (0.64) ACHELMNACYP3A4CYP1A2CYP2D6
SCHEMBL14387221 0.76 ACHE (0.52) ACHELMNACYP3A4CYP1A2CYP2D6
SCHEMBL10747649 0.76 ACHE (0.59) ACHELMNACYP3A4CYP1A2CYP2D6
SCHEMBL1753213 0.76 ACHE (0.54) ACHELMNACYP3A4CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4677106-A ANTIDEPRESSANTS SANOFI (FR) 1987-06-30 US disclosed
US-4576946-A ANTIDEPRESSANT SANOFI (FR) 1986-03-18 US disclosed
US-4514397-A Derivatives of 4-methyl 6-phenyl pyridazine active on the central nervous system SANOFI (FR) 1985-04-30 US disclosed