Bromide

Bromide

SCHEMBL10749029

Br.CCOC(=O)Nc1cccc(-c2csc(N=C(N)N)n2)c1

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 13/20 0.60
ATP4B P51164 13/20 0.60
HDAC3 O15379 4/20 0.57
HDAC1 Q13547 3/20 0.57
HDAC2 Q92769 3/20 0.57
HDAC10 Q969S8 2/20 0.57
HDAC8 Q9BY41 2/20 0.57
HDAC6 Q9UBN7 2/20 0.57
HDAC4 P56524 1/20 0.57
HDAC7 Q8WUI4 1/20 0.57
HDAC11 Q96DB2 1/20 0.57
HDAC9 Q9UKV0 1/20 0.57
HDAC5 Q9UQL6 1/20 0.57
NCOR2 Q9Y618 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL10750011 0.87 MAPT (0.58) ATP4AATP4B
Bromide SCHEMBL10753076 0.82 HDAC3 (0.65) ATP4AATP4BHDAC3HDAC1HDAC2
Bromide SCHEMBL10749032 0.82 HDAC3 (0.67) HDAC3HDAC1HDAC2HDAC10HDAC8
Bromide SCHEMBL10726966 0.81 HDAC3 (0.69) HDAC3HDAC1HDAC2HDAC10HDAC8
SCHEMBL10810745 0.81 HDAC3 (0.66) ATP4AATP4BHDAC3HDAC1HDAC2
SCHEMBL10812025 0.80 HDAC3 (0.68) HDAC3HDAC1HDAC2HDAC10HDAC8
SCHEMBL11148430 0.80 HDAC3 (0.70) HDAC3HDAC1HDAC2HDAC10HDAC8
Bromide SCHEMBL10753066 0.79 HDAC3 (0.57) HDAC3HDAC1HDAC2HDAC10HDAC8
SCHEMBL10810738 0.78 HDAC3 (0.58) HDAC3HDAC1HDAC2HDAC10HDAC8
Bromide SCHEMBL827268 0.76 ATP4A (1.00) ATP4AATP4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4645841-A ANTIULCER AGENTS ISTITUTO DE ANGELI, S.P.A. (IT) 1987-02-24 US disclosed
US-4548944-A ANTIULCER, ANTISECRETORY AGENTS ISTITUTO DE ANGELI S.P.A. (IT) 1985-10-22 US disclosed