SCHEMBL10749685

SCHEMBL10749685

COc1cc2c(cc1SC)CCN(C)CC2c1ccccc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.78
CYP3A4 P08684 2/20 0.78
DRD1 P21728 14/20 0.59
HSD17B10 Q99714 4/20 0.59
THPO P40225 2/20 0.59
MAPK1 P28482 2/20 0.59
HIF1A Q16665 1/20 0.59
MTOR P42345 1/20 0.59
DRD2 P14416 4/20 0.58
KDM4E B2RXH2 1/20 0.58
MAPT P10636 1/20 0.58
BLM P54132 1/20 0.58
PMP22 Q01453 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
HTR2A P28223 2/20 0.55
DRD5 P21918 4/20 0.55
CYP1A2 P05177 3/20 0.55
TSHR P16473 3/20 0.55
NFKB1 P19838 1/20 0.55
CYP2C19 P33261 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10745747 0.99 CYP2D6 (0.76) CYP2D6CYP3A4DRD1HSD17B10THPO
Trepipam SCHEMBL11704977 0.88 CYP2D6 (1.00) CYP2D6CYP3A4DRD1HSD17B10THPO
Trepipam SCHEMBL29374758 0.88 CYP2D6 (1.00) CYP2D6CYP3A4DRD1HSD17B10THPO
Hydrochloric Acid SCHEMBL10345632 0.88 CYP2D6 (0.73) CYP2D6CYP3A4DRD1HSD17B10THPO
SCHEMBL11939886 0.83 CYP2D6 (0.81) CYP2D6CYP3A4DRD1HSD17B10THPO
SCHEMBL11112777 0.83 CYP2D6 (0.81) CYP2D6CYP3A4DRD1HSD17B10THPO
SCHEMBL10345387 0.83 CYP2D6 (0.81) CYP2D6CYP3A4DRD1HSD17B10THPO
SCHEMBL10745139 0.83 DRD1 (0.77) CYP2D6CYP3A4DRD1HSD17B10THPO
SCHEMBL10746175 0.82 CYP3A4 (0.53) CYP2D6CYP3A4DRD1HSD17B10THPO
Bromide SCHEMBL10744885 0.82 KDM4E (0.77) CYP2D6CYP3A4DRD1HSD17B10THPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0244088-A2 1-Phenyl-3-benzazepine compounds and medicaments containing these compounds for treating gastrointestinal motility disorders SMITHKLINE BEECHAM CORPORATION (US) 1987-11-04 EP disclosed