SCHEMBL10766870

SCHEMBL10766870

C=CCn1cccc(C#N)c1=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.61
ALDH1A1 P00352 8/20 0.61
HPGD P15428 7/20 0.61
GAA P10253 5/20 0.61
GLA P06280 2/20 0.61
RCE1 Q9Y256 1/20 0.61
ALOX12 P18054 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.51
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
NPC1 O15118 8/20 0.44
KMT2A Q03164 5/20 0.44
RAB9A P51151 7/20 0.43
MEN1 O00255 3/20 0.43
S1PR2 O95136 1/20 0.41
S1PR4 O95977 1/20 0.41
ESR1 P03372 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5574433 0.85 ALDH1A1 (0.48) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL10462174 0.81 KDM4E (0.40) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL27397322 0.77 KDM4E (0.50) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL11833611 0.77 STAT3 (0.51) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL83810 0.75 KDM4E (0.41) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL7037632 0.74 EGLN1 (0.51) ALDH1A1NPC1KMT2ARAB9AMEN1
SCHEMBL9356553 0.73 ALDH1A1 (0.50) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL13448507 0.73 GRM2 (0.43) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL26750149 0.73 GRM2 (0.39) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL25316781 0.72 NPC1 (0.49) KDM4EALDH1A1HPGDGAAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4645766-A 1,2-dihydro-2-oxo-3-hydroxymethyl pyridines, compositions and use THE UPJOHN COMPANY (US) 1987-02-24 US disclosed
US-4108630-A 1-Alkylpyrid-2-ones ROHM AND HAAS COMPANY (US) 1978-08-22 US disclosed
US-4038065-A 1-ALKYLPYRID-2-ONE ROHM AND HAAS COMPANY (US) 1977-07-26 US disclosed