SCHEMBL10767151

SCHEMBL10767151

COC(=O)C1=C(CF)NC(C)=C(C(=O)OC(C)C)C1c1cc(OC)ccc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 8/20 0.51
CYP3A4 P08684 7/20 0.51
CYP2C9 P11712 7/20 0.51
CYP2C19 P33261 7/20 0.51
ADORA3 P0DMS8 6/20 0.51
LMNA P02545 6/20 0.51
KMT2A Q03164 6/20 0.51
CACNA1C Q13936 5/20 0.51
MAPT P10636 5/20 0.51
SCN5A Q14524 4/20 0.51
CACNA1F O60840 4/20 0.51
CACNA1D Q01668 4/20 0.51
CACNA1S Q13698 4/20 0.51
CYP2D6 P10635 4/20 0.51
HIF1A Q16665 4/20 0.51
ABCB11 O95342 3/20 0.51
KCNH2 Q12809 3/20 0.51
TSHR P16473 3/20 0.51
NFKB1 P19838 3/20 0.51
THPO P40225 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7425671 0.87 CYP1A2 (0.69) CYP1A2CYP3A4CYP2C9CYP2C19ADORA3
SCHEMBL10766752 0.86 KDM4E (0.48) CYP1A2CYP3A4CYP2C9CYP2C19ADORA3
SCHEMBL7438846 0.84 CYP1A2 (0.56) CYP1A2CYP3A4CYP2C9CYP2C19ADORA3
SCHEMBL7434480 0.83 CYP1A2 (0.58) CYP1A2CYP3A4CYP2C9CYP2C19ADORA3
SCHEMBL7434250 0.82 CYP1A2 (0.56) CYP1A2CYP3A4CYP2C9CYP2C19ADORA3
SCHEMBL7427392 0.81 ADORA3 (0.56) CYP1A2CYP3A4CYP2C9CYP2C19ADORA3
SCHEMBL7266447 0.81 ADORA3 (0.45) CYP1A2CYP3A4CYP2C9CYP2C19ADORA3
SCHEMBL10767938 0.80 CYP1A2 (0.54) CYP1A2CYP3A4CYP2C9CYP2C19ADORA3
SCHEMBL7426393 0.80 ADORA3 (0.54) CYP1A2CYP3A4CYP2C9CYP2C19ADORA3
SCHEMBL7381462 0.79 CYP1A2 (0.69) CYP1A2CYP3A4CYP2C9CYP2C19ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0225175-A2 Dihydropyridine derivatives, processes for their preparation and pharmaceutical compositions thereof FISONS plc (GB) 1987-06-10 EP claimed
EP-0225175-A2 Dihydropyridine derivatives, processes for their preparation and pharmaceutical compositions thereof FISONS plc (GB) 1987-06-10 EP disclosed