SCHEMBL1077045

SCHEMBL1077045

O=C1C=CONN1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL345261 0.59
SCHEMBL11816980 0.59 GSK3A (0.41)
SCHEMBL4585773 0.56
SCHEMBL28390358 0.56
SCHEMBL2519473 0.56
SCHEMBL279748 0.56
Hydrochloric Acid SCHEMBL2519134 0.54
SCHEMBL699281 0.54
SCHEMBL1952488 0.51
SCHEMBL616019 0.50

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 117 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6013686-A A BLOWING AGENT CONCENTRATE FOR PRODUCING FOAMED PARTS UPON MOLDING, COMPRISES A POLYCARBONATE-POLYESTER COPOLYMER, THE MONOMER UNITS DERIVED FROM DIHYDRIC PHENOL AND DICARBOXYLIC ACID, BLOWING AGENT WITH SELECTED GAS GENERATION TEMPERATURE GENERAL ELECTRIC COMPANY (US) 2000-01-11 US claimed
EP-0601783-B1 Blowing agent concentrate GEN ELECTRIC (US) 1999-04-14 EP claimed
EP-0385092-A2 Foamable engineering thermoplastic compositions GENERAL ELECTRIC COMPANY (US) 1990-09-05 EP claimed
US-4904702-A Foamable engineering thermoplastic compositions GENERAL ELECTRIC COMPANY (US) 1990-02-27 US claimed
US-4683247-A Foamable thermoplastic compositions, foamed articles and foaming method based on pre-compounded nucleating agent-resin concentrate GENERAL ELECTRIC COMPANY (US) 1987-07-28 US claimed
US-4587272-A Foamable polycarbonate compositions, articles and methods GENERAL ELECTRIC COMPANY (US) 1986-05-06 US claimed
EP-0158266-A2 Foamable polycarbonate compositions, articles and methods GENERAL ELECTRIC COMPANY (US) 1985-10-16 EP claimed
US-4544677-A IMPACT STRENGTH GENERAL ELECTRIC COMPANY (US) 1985-10-01 US claimed
US-4334030-A INJECTION MOLDABLE CONCENTRATES CONTAINING AMIDE DERIVATIVES OF AZODICARBOXYLIC ACID AND A DIHYDROOXADIAZINONE AS BLOWING AGENTS GENERAL ELECTRIC COMPANY (US) 1982-06-08 US claimed
US-4163037-A USING A DIHYDROOXADIAZINONE BLOWING AGENT, INJECTION MOLDING GENERAL ELECTRIC COMPANY (US) 1979-07-31 US claimed
US-4160088-A HALOGENATION OF KETONE, ALKANOL, HYDROLYSIS GENERAL ELECTRIC COMPANY (US) 1979-07-03 US claimed
US-4158094-A BLOWING AGENTS GENERAL ELECTRIC COMPANY (US) 1979-06-12 US claimed
US-4105848-A Process for the production of dihydrooxadiazinone compounds GENERAL ELECTRIC COMPANY (US) 1978-08-08 US claimed
US-4097425-A POLYCARBONATES, POLYESTERS, SUBSTITUTED 3,6-DIHYDRO-1,3,4-OXDIAZIN-2-ONE GENERAL ELECTRIC COMPANY (US) 1978-06-27 US claimed
JP-2283734-A None JP disclosed
EP-4541791-A1 DIHYDROOXADIAZINONE COMPOUND AND PHARMACEUTICAL USE THEREOF Japan Tobacco Inc. (JP) 2025-04-23 EP disclosed
US-12258323-B2 Dihydrooxadiazinones BAYER AKTIENGESELLSCHAFT (DE) 2025-03-25 US disclosed
US-4097671-A 5-PHENYL-3,6-DIHYDRO-1,3,4-OXADIAZIN-2-ONE, THERMOPLASTIC POLYMER BLOWING AGENT GENERAL ELECTRIC COMPANY (US) 1978-06-27 US disclosed
US-4097671-A 5-PHENYL-3,6-DIHYDRO-1,3,4-OXADIAZIN-2-ONE, THERMOPLASTIC POLYMER BLOWING AGENT GENERAL ELECTRIC COMPANY (US) 1978-06-27 US disclosed
US-4097671-A 5-PHENYL-3,6-DIHYDRO-1,3,4-OXADIAZIN-2-ONE, THERMOPLASTIC POLYMER BLOWING AGENT GENERAL ELECTRIC COMPANY (US) 1978-06-27 US disclosed