SCHEMBL10778149

SCHEMBL10778149

CC(=Cc1ccccc1C1C(C(=O)O)=C(C)NC(C)=C1C(=O)O)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.42
LMNA P02545 2/20 0.41
CYP3A4 P08684 2/20 0.41
ADORA3 P0DMS8 2/20 0.41
CYP2C9 P11712 2/20 0.41
TBXAS1 P24557 2/20 0.41
CYP2C19 P33261 2/20 0.41
KCNH2 Q12809 2/20 0.41
NR1I2 O75469 2/20 0.41
HTT P42858 1/20 0.41
PGR P06401 1/20 0.41
SLC6A2 P23975 1/20 0.41
DRD3 P35462 1/20 0.41
OPRK1 P41145 1/20 0.41
PDE4D Q08499 1/20 0.41
CACNA1B Q00975 12/20 0.40
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
MAPK1 P28482 2/20 0.38
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10778133 1.00 AKR1C3 (0.42) AKR1C3LMNACYP3A4ADORA3CYP2C9
SCHEMBL10778144 1.00 AKR1C3 (0.42) AKR1C3LMNACYP3A4ADORA3CYP2C9
SCHEMBL9524555 0.85 BRD4 (0.41) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9524567 0.85 BRD4 (0.41) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9524561 0.85 BRD4 (0.41) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL10772083 0.85 ADORA3 (0.49) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9680643 0.85 ADORA3 (0.60) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9680632 0.85 ADORA3 (0.60) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9680646 0.85 ADORA3 (0.60) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL10772073 0.85 ADORA3 (0.49) LMNACYP3A4ADORA3CYP2C9TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0226271-A1 1,4-Dihydropyridine compounds and their preparation and pharmaceutical formulation GLAXO S.p.A. (IT) 1987-06-24 EP disclosed