SCHEMBL1078360

SCHEMBL1078360

C=CCc1cccc2c1N=N[N]2

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.42
GABRB2 P47870 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.35
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
KMT2A Q03164 5/20 0.33
ALDH1A1 P00352 5/20 0.33
MEN1 O00255 4/20 0.33
GAA P10253 3/20 0.33
LMNA P02545 2/20 0.33
AKR1B1 P15121 1/20 0.33
MAPT P10636 3/20 0.32
MAPK1 P28482 1/20 0.32
KDM4E B2RXH2 3/20 0.31
HSD17B10 Q99714 3/20 0.31
CASP1 P29466 1/20 0.31
ALOX12 P18054 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5603693 0.73 GRM5 (0.33) ALDH1A1GAAKDM4E
SCHEMBL1079897 0.71 GABRA1 (0.42) GABRA1GABRB2L3MBTL1ADRA2AADRA2B
SCHEMBL7608071 0.70 GABRA1 (0.49) GABRA1GABRB2L3MBTL1ADRA2AADRA2B
SCHEMBL5600974 0.69 CNR2 (0.35) ALDH1A1
SCHEMBL5824091 0.67 GABRA1 (0.58) GABRA1GABRB2L3MBTL1ADRA2AADRA2B
SCHEMBL173300 0.66 GABRA1 (0.56) GABRA1GABRB2L3MBTL1ADRA2AADRA2B
SCHEMBL29763626 0.66 GABRA1 (0.56) GABRA1GABRB2L3MBTL1ADRA2AADRA2B
SCHEMBL10797073 0.66 GABRA1 (0.52) GABRA1GABRB2L3MBTL1ADRA2AADRA2B
SCHEMBL31619949 0.65 GABRA1 (0.56) GABRA1GABRB2L3MBTL1KMT2AALDH1A1
SCHEMBL18136 0.65 GABRA1 (0.56) GABRA1GABRB2L3MBTL1ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0408509-B1 Substituted benzonitriles CIBA GEIGY AG (CH) 1996-03-06 EP claimed
EP-2448926-A1 FLAVIN DERIVATIVES Biorelix, Inc. (US) 2012-05-09 EP disclosed
WO-2011008247-A1 FLAVIN DERIVATIVES BIORELIX, INC. (US) 2011-01-20 WO disclosed
US-5073574-A TETRAZOLYL SUBSTITUTED BENZONITRILES AND ANTI-TUMOR USE THEREOF CIBA-GEIGY CORPORATION (US) 1991-12-17 US disclosed