SCHEMBL10795290

SCHEMBL10795290

S=C1c2nc[nH]c2N(Cc2ccc(Cl)cc2)C2=NCCN12

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.50
HTT P42858 4/20 0.43
GAA P10253 1/20 0.40
GFER P55789 1/20 0.40
TP53 P04637 2/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.35
CLPP Q16740 1/20 0.35
ACP1 P24666 1/20 0.34
SOS1 Q07889 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
LMNA P02545 3/20 0.33
DBH P09172 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10795495 0.86 TSHR (0.50) TSHRHTTGAAGFERTP53
SCHEMBL10795586 0.86 TSHR (0.57) TSHRHTTGAAGFERTP53
Hydrochloric Acid SCHEMBL11069993 0.85 TSHR (0.56) TSHRHTTGAAGFERTP53
SCHEMBL10800156 0.80 TSHR (0.52) TSHRHTTGAATP53KMT2A
SCHEMBL14540610 0.77 TSHR (0.43) TSHRHTTKMT2AMEN1CLPP
SCHEMBL11066311 0.76 HTT (0.51) TSHRHTTGAAGFERTP53
SCHEMBL10795826 0.75 GAA (0.52) TSHRHTTGAAGFERTP53
SCHEMBL11064805 0.75 TSHR (0.47) TSHRGAAGFERTP53KMT2A
SCHEMBL11163356 0.72 TSHR (0.57) TSHRHTTGAAGFERTP53
Water SCHEMBL10795500 0.71 TSHR (0.56) TSHRHTTGAAGFERTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4642345-A BRONCHODILATOR AGENTS MEAD JOHNSON & COMPANY (US) 1987-02-10 US disclosed
US-4489078-A Diazaheterocyclopurines used as anti-broncho spasmatics and vasodilators MEAD JOHNSON & COMPANY (US) 1984-12-18 US disclosed
US-4404380-A BRONCHODILATORS, MEDIATOR RELEASE INHIBITORS, PHOSPHODIESTERASE INHIBITORS, AND VASODILATORS MEAD JOHNSON & COMPANY (US) 1983-09-13 US disclosed
US-4366156-A Antiallergic methods using diazaheterocyclopurines MEAD JOHNSON & COMPANY (US) 1982-12-28 US disclosed