SCHEMBL10797368

SCHEMBL10797368

N#Cc1ccc(S(=O)(=O)C2CCCNC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
APLNR P35414 2/20 0.45
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
KCNH2 Q12809 1/20 0.40
PTGS2 P35354 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CCR6 P51684 3/20 0.39
CYP19A1 P11511 1/20 0.39
KDM1A O60341 1/20 0.37
MMP1 P03956 1/20 0.37
MMP8 P22894 1/20 0.37
MMP13 P45452 1/20 0.37
THRB P10828 1/20 0.36
CXCR2 P25025 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10794480 0.98 APLNR (0.44) APLNRDRD2DRD3HTR2AHTR2C
SCHEMBL2581906 0.82 HTR2A (0.47) HTR2AHTR2CKCNH2PTGS2CA12
SCHEMBL10795117 0.81 APLNR (0.47) APLNRCXCR2
SCHEMBL10795010 0.81 APLNR (0.47) APLNRCA2MMP1MMP8MMP13
SCHEMBL10799201 0.81 APLNR (0.47) APLNRDRD2HTR2AHTR2CKCNH2
SCHEMBL10794767 0.81 APLNR (0.47) APLNRPTGS2MMP1MMP8MMP13
SCHEMBL10794469 0.81 APLNR (0.47) APLNRMMP1MMP8MMP13CXCR2
SCHEMBL10795613 0.81 APLNR (0.47) APLNRMMP1MMP8MMP13CXCR2
SCHEMBL5209868 0.81 KCNH2 (0.46) HTR2AHTR2CKCNH2PTGS2CA12
SCHEMBL711807 0.81 APLNR (0.50) APLNRHTR2AHTR2CKCNH2MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4642348-A ANTIARRHYTHMIA AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1987-02-10 US disclosed
US-4593102-A N-[(amino)alkyl]-1-pyrrolidine, 1-piperidine and 1-homopiperidinecarboxamides (and thiocarboxamides) with sulfur linked substitution in the 2, 3 or 4-position A. H. ROBINS COMPANY, INC. (US) 1986-06-03 US disclosed
EP-0160436-A2 N-[(Amino)Alkyl]-1-pyrrolidine, 1-piperidine and 1-homopiperidinecarboxamides (and thiocarboxamides) with sulphur linked substitution in the 2, 3 or 4-position A.H. ROBINS COMPANY, INCORPORATED (US) 1985-11-06 EP disclosed