SCHEMBL10813992

SCHEMBL10813992

OC(Cn1ccnc1)(Cn1cncn1)c1ccc(Cl)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OGG1 O15527 1/20 0.54
CYP27B1 O15528 1/20 0.52
CYP3A4 P08684 8/20 0.49
CYP2C9 P11712 4/20 0.49
CYP2C19 P33261 4/20 0.49
LMNA P02545 1/20 0.49
HSP90AA1 P07900 1/20 0.49
CYP19A1 P11511 1/20 0.49
CYP11B1 P15538 1/20 0.49
CYP11B2 P19099 1/20 0.49
ADRA1A P35348 1/20 0.49
CYP51A1 Q16850 1/20 0.49
PTGS2 P35354 1/20 0.48
ADRA2C P18825 2/20 0.44
PDCD1 Q15116 1/20 0.43
CD274 Q9NZQ7 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2D6 P10635 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8057057 0.89 CYP3A4 (0.59) OGG1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL9665470 0.83 OGG1 (0.61) OGG1CYP27B1CYP3A4CYP2C9CYP2C19
SCHEMBL10917880 0.83 OGG1 (0.61) OGG1CYP27B1CYP3A4CYP2C9CYP2C19
SCHEMBL10916395 0.83 OGG1 (0.61) OGG1CYP27B1CYP3A4CYP2C9CYP2C19
SCHEMBL11119666 0.83 CYP3A4 (0.52) OGG1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL8757356 0.82 CYP3A4 (0.49) OGG1CYP27B1CYP3A4CYP2C9CYP2C19
SCHEMBL11372412 0.82 OGG1 (0.60) OGG1CYP27B1CYP3A4CYP2C9CYP2C19
SCHEMBL10916378 0.82 OGG1 (0.60) OGG1CYP27B1CYP3A4CYP2C9CYP2C19
SCHEMBL10916373 0.82 OGG1 (0.60) OGG1CYP27B1CYP3A4CYP2C9CYP2C19
SCHEMBL9308406 0.82 CYP3A4 (0.51) OGG1CYP3A4CYP2C9CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0126581-B1 ANTIFUNGAL TRIAZOLE DERIVATIVES Pfizer Limited (GB) 1987-06-03 EP disclosed
EP-0044605-B1 FUNGICIDAL BIS-AZOLYL COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-02-12 EP disclosed
US-4554286-A Antifungal 1-triazolyl-2-aryl-3-(5-trifluoromethylimidazol-1-yl)propan-2-ol derivatives PFIZER INC. (US) 1985-11-19 US disclosed
US-4523019-A INTERMEDIATE FOR FUNGICIDE AND PLANT GROWTH REGULATOR IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-06-11 US disclosed
EP-0126581-A1 Antifungal triazole derivatives Pfizer Limited (GB) 1984-11-28 EP disclosed
EP-0111658-A2 1,3-Dihalopropan-2-ols IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-06-27 EP disclosed
US-4416682-A 1,3-Bis(azolyl)propanols as fungicides and plant growth regulators IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-11-22 US disclosed
EP-0044605-A1 Fungicidal bis-azolyl compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-01-27 EP disclosed