SCHEMBL10817029

SCHEMBL10817029

Cc1cnc(Nc2ccccc2)c([N+](=O)[O-])c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.56
PIN1 Q13526 1/20 0.55
TDP1 Q9NUW8 3/20 0.53
MAPT P10636 4/20 0.49
MAPK1 P28482 4/20 0.49
POLB P06746 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
ALDH1A1 P00352 2/20 0.48
L3MBTL1 Q9Y468 5/20 0.47
CASP7 P55210 1/20 0.47
JAK2 O60674 1/20 0.47
GSK3A P49840 2/20 0.47
AURKA O14965 1/20 0.47
LMNA P02545 3/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12100780 0.89 RAB9A (0.56) GSK3BTDP1MAPTMAPK1POLB
SCHEMBL1699272 0.84 MAPT (0.53) GSK3BTDP1MAPTMAPK1POLB
SCHEMBL6386431 0.84 TDP1 (0.44) GSK3BPIN1TDP1MAPTMAPK1
SCHEMBL29695587 0.84 TDP1 (0.73) GSK3BPIN1TDP1MAPTMAPK1
SCHEMBL13506718 0.82 GSK3B (0.56) GSK3BPIN1TDP1MAPTMAPK1
SCHEMBL10138757 0.82 GSK3B (0.56) GSK3BPIN1TDP1MAPTMAPK1
SCHEMBL10810189 0.82 JAK2 (0.58) GSK3BPIN1TDP1MAPTMAPK1
SCHEMBL1858862 0.81 KMT2A (0.56) TDP1MAPTMAPK1POLBALDH1A1
SCHEMBL1624745 0.80 TDP1 (0.49) GSK3BTDP1MAPTMAPK1POLB
SCHEMBL31717653 0.79 MAPK1 (0.78) GSK3BPIN1TDP1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4698430-A ANTIDEPRESSANT A. H. ROBINS COMPANY, INC. (US) 1987-10-06 US disclosed
US-4558132-A ANTIDEPRESSANTS A. H. ROBINS COMPANY, INCORPORATED (US) 1985-12-10 US disclosed
EP-0099614-A2 Nitro, amino and aroylamino-N-phenylpyridinamines and their use in a process for preparing pyrido(1,4)benzodiazapines A.H. ROBINS COMPANY, INCORPORATED (US) 1984-02-01 EP disclosed