SCHEMBL10822232

SCHEMBL10822232

CC(C)(C)N(C(=O)O)[C@@H](C(=O)O)c1ccc(O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.41
ESR1 P03372 10/20 0.38
ESR2 Q92731 8/20 0.38
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
CYP3A4 P08684 4/20 0.35
ALDH1A1 P00352 3/20 0.35
BLM P54132 1/20 0.35
CYP2C9 P11712 3/20 0.35
CYP2C19 P33261 2/20 0.35
HSD17B10 Q99714 1/20 0.35
APP P05067 1/20 0.35
TDP1 Q9NUW8 2/20 0.34
LMNA P02545 2/20 0.34
CYP1A2 P05177 1/20 0.34
PGR P06401 1/20 0.34
CHRM2 P08172 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
AR P10275 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1443507 0.85 ESR1 (0.44) ESR1ESR2KMT2A
SCHEMBL28637927 0.84 BRD4 (0.41) CYP3A4BLMCYP2C9CYP2C19HSD17B10
SCHEMBL2429212 0.82 ESR1 (0.42) SRCESR1ESR2PDCD1CD274
SCHEMBL1448846 0.82 ESR1 (0.42) SRCESR1ESR2PDCD1CD274
SCHEMBL28656346 0.81 NPSR1 (0.46) ALDH1A1TDP1CYP1A2MAPTPTGS1
SCHEMBL17764981 0.81 NR1H2 (0.40) ALDH1A1CYP2C9CYP2C19LMNACYP1A2
SCHEMBL17764980 0.81 NR1H2 (0.40) ALDH1A1CYP2C9CYP2C19LMNACYP1A2
SCHEMBL7647994 0.78 NPY5R (0.46) ESR1ESR2PDCD1CD274CYP3A4
SCHEMBL16633588 0.78 ESR1 (0.43) ESR1ESR2PDCD1CD274CYP3A4
SCHEMBL10822196 0.78 ESR1 (0.34) SRCESR1ESR2PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4604386-A CONTROL OF GRAMPOSITIVE BACTERIA ELI LILLY AND COMPANY (US) 1986-08-05 US disclosed
EP-0168222-A2 3-(Alkynylalkyloxy) Cephalosporins ELI LILLY AND COMPANY (US) 1986-01-15 EP disclosed