SCHEMBL28656346

SCHEMBL28656346

COc1ccc([C@@H](C(=O)O)N(C(=O)O)C(C)(C)C)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.46
LDHA P00338 1/20 0.44
BMP1 P13497 1/20 0.43
AKR1C3 P42330 6/20 0.43
AKR1C2 P52895 6/20 0.43
PTGS2 P35354 3/20 0.43
PTGS1 P23219 3/20 0.43
CYP1A2 P05177 2/20 0.43
CDC42 P60953 1/20 0.43
RAC1 P63000 1/20 0.43
TSHR P16473 1/20 0.43
SLC22A6 Q4U2R8 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
ACP3 P15309 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 1/20 0.41
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10822232 0.81 SRC (0.41) PTGS1CYP1A2ALDH1A1MAPTTDP1
SCHEMBL836811 0.80 NPY5R (0.49) NPSR1BMP1AKR1C3AKR1C2PTGS2
SCHEMBL17603763 0.80 BMP1 (0.43) NPSR1LDHABMP1ACP3L3MBTL1
SCHEMBL1673370 0.80 NPSR1 (0.43) NPSR1BMP1AKR1C3AKR1C2PTGS2
SCHEMBL28637927 0.80 BRD4 (0.41) CYP1A2TSHRMAPT
SCHEMBL2091000 0.80 LDHA (0.49) NPSR1LDHAAKR1C3AKR1C2PTGS2
SCHEMBL6349734 0.79 TAS1R3 (0.43) NPSR1LDHABMP1AKR1C3AKR1C2
SCHEMBL1673386 0.79 ALOX5 (0.43) NPSR1BMP1AKR1C3AKR1C2PTGS2
SCHEMBL5862818 0.77 BMP1 (0.41) NPSR1LDHABMP1L3MBTL1ALDH1A1
SCHEMBL11441436 0.77 LDHA (0.50) NPSR1LDHAAKR1C3AKR1C2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107531653-B Novel difluoroketoamide derivatives 豪夫迈·罗氏有限公司 2021-10-19 CN disclosed