SCHEMBL10828239

SCHEMBL10828239

CC1(C)C(=O)Nc2c(O)cccc21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 4/20 0.61
PDK4 Q16654 3/20 0.59
PDK1 Q15118 1/20 0.59
PDK3 Q15120 1/20 0.59
CNR1 P21554 1/20 0.41
HTT P42858 1/20 0.41
GPR35 Q9HC97 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
PGR P06401 5/20 0.38
EPHX2 P34913 1/20 0.36
NPSR1 Q6W5P4 3/20 0.36
LMNA P02545 2/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.34
CYP1A2 P05177 1/20 0.34
PARP1 P09874 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2264510 0.78 PDK2 (0.62) PDK2PDK4PDK1PDK3CNR1
SCHEMBL2269040 0.77 PDK2 (0.61) PDK2PDK4PDK1PDK3PGR
SCHEMBL3138211 0.77 PDK2 (0.61) PDK2PDK4PDK1PDK3CNR1
SCHEMBL31117008 0.77 PDK2 (0.61) PDK2PDK4PDK1PDK3CNR1
SCHEMBL31032206 0.77 PDK2 (0.56) PDK2PDK4PDK1PDK3CNR1
SCHEMBL10470225 0.76 PDK2 (0.59) PDK2PDK4PDK1PDK3CNR1
SCHEMBL10828347 0.74 PDK2 (0.57) PDK2PDK4PDK1PDK3KMT2A
SCHEMBL10915783 0.73 PGR (0.41) PDK2KMT2AMEN1PGR
SCHEMBL10482937 0.72 MEN1 (0.36) PDK2PDK4CNR1HTTGPR35
SCHEMBL3150359 0.71 PDK2 (0.52) PDK2PDK4PDK1PDK3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4622336-A ANALGESICS SANDOZ LTD. (CH) 1986-11-11 US disclosed
WO-1983002610-A1 DERIVATIVES OF 3,3-DIALKYL-INDOLIN AND OF 3,3-ALKYLENE-INDOLIN, METHOD FOR PRODUCING THEM AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM SANDOZ AG (CH) 1983-08-04 WO disclosed