SCHEMBL10828697

SCHEMBL10828697

CCOC(=O)CC[C@H](NC(=O)c1ccc(N(CCF)Cc2ccc3nc(N)nc(O)c3c2)cc1)C(=O)OCC

nearest known ligand 0.57

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DHFR P00374 8/20 0.53
TYMS P04818 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10828701 1.00 DHFR (0.53) DHFRTYMS
SCHEMBL10828966 0.90 DHFR (0.59) DHFRTYMS
SCHEMBL10828968 0.90 DHFR (0.59) DHFRTYMS
SCHEMBL10828741 0.89 DHFR (0.50) DHFRTYMS
SCHEMBL10828695 0.89 DHFR (0.59) DHFRTYMS
SCHEMBL10828745 0.89 DHFR (0.50) DHFRTYMS
SCHEMBL10828694 0.89 DHFR (0.59) DHFRTYMS
SCHEMBL14028320 0.88 DHFR (0.57) DHFRTYMS
SCHEMBL10828954 0.88 DHFR (0.48) DHFRTYMS
SCHEMBL10828952 0.88 DHFR (0.48) DHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4564616-A Anti-cancer quinazoline derivatives NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1986-01-14 US disclosed
EP-0031237-B1 QUINAZOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTI-CANCER AGENTS NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1984-10-17 EP disclosed
US-4447608-A ANTITUMOR AGENTS NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1984-05-08 US disclosed
EP-0031237-A1 Quinazoline derivatives, processes for their preparation, compositions containing them and their use as anti-cancer agents NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1981-07-01 EP disclosed