SCHEMBL10837697

SCHEMBL10837697

COc1ccc2c3c1CCCC3C(=O)CC2

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.44
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
PARP1 P09874 1/20 0.38
NQO2 P16083 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9312311 0.80 BRD4 (0.44) ADRA1AGAAPARP1
SCHEMBL10468029 0.77 PARP1 (0.42) GAAPARP1
SCHEMBL10468977 0.71 BRD4 (0.44) GAAPARP1
SCHEMBL10836480 0.71 TLR4 (0.38) ADRA1A
Hydrochloric Acid SCHEMBL10836770 0.71 ADRA1A (0.51) ADRA1A
SCHEMBL10838426 0.70 ADRA1A (0.42) ADRA1ANQO2MTNR1AMTNR1B
SCHEMBL15911203 0.69 ADRA1A (0.49) ADRA1AKDM4EALDH1A1GLAGAA
Hydrochloric Acid SCHEMBL10838511 0.69 ADRA1A (0.43) ADRA1A
Hydrochloric Acid SCHEMBL10838208 0.69 ADRA1A (0.43) ADRA1A
Hydrochloric Acid SCHEMBL10836525 0.69 ADRA1A (0.43) ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4564698-A Biologically-active tricyclic amines AKZO N.V. (NL) 1986-01-14 US disclosed
EP-0041293-B1 BIOLOGICALLY-ACTIVE TRICYCLIC AMINES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AKZO N.V. (NL) 1984-03-14 EP disclosed
WO-1981003490-A1 BIOLOGICALLY-ACTIVE TRICYCLIC AMINES,METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AKZO NV (NL) 1981-12-10 WO disclosed
EP-0041293-A1 Biologically-active tricyclic amines, methods for their preparation and pharmaceutical compositions containing same AKZO N.V. (NL) 1981-12-09 EP disclosed