SCHEMBL10838751

SCHEMBL10838751

COc1ccc(C(=O)CCCl)c2c1NC(=O)CC2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
HSD17B10 Q99714 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
STAT6 P42226 1/20 0.35
FLI1 Q01543 1/20 0.34
EWSR1 Q01844 1/20 0.34
HTR2A P28223 3/20 0.34
HTR2C P28335 3/20 0.34
HTR2B P41595 3/20 0.34
ADRB3 P13945 1/20 0.34
KDM4E B2RXH2 3/20 0.34
HPGD P15428 3/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
CRBN Q96SW2 2/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
PDE4D Q08499 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8920419 0.90 FLI1 (0.38) ALDH1A1HSD17B10FLI1EWSR1ADRB3
SCHEMBL8921162 0.82 MAPT (0.43) ALDH1A1HSD17B10ADRB3KDM4EHPGD
SCHEMBL11865700 0.82 KDM4E (0.37) ALDH1A1HSD17B10CYP1A2CYP3A4CYP2C9
SCHEMBL10541813 0.82 HTR2A (0.39) ALDH1A1HSD17B10CYP1A2CYP3A4CYP2C9
SCHEMBL11874083 0.80 ADRB3 (0.37) ALDH1A1HSD17B10CYP1A2CYP3A4CYP2C9
SCHEMBL11704700 0.79 ADRB3 (0.37) ALDH1A1HSD17B10FLI1EWSR1ADRB3
SCHEMBL11861861 0.79 ADRB2 (0.40) ALDH1A1HSD17B10CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL11861584 0.78 ADRB3 (0.36) ALDH1A1HSD17B10FLI1EWSR1ADRB3
SCHEMBL9385137 0.77 ADRB3 (0.40) ALDH1A1ADRB3KDM4EHPGDGLA
SCHEMBL9384972 0.77 ADRB3 (0.40) ALDH1A1ADRB3KDM4EHPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4619932-A CENTRAL NERVOUS SYSTEM CONTROLLERS; ANTI-SCHIZOPHRENIA AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-10-28 US disclosed
US-4567187-A CENTRAL NERVOUS SYSTEM OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-01-28 US disclosed
US-4460593-A Carbostyril derivatives, and central nervous system controlling agents containing the carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-07-17 US disclosed
US-4455422-A ANTIHISTAMINES, CNS CONTROLLERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-19 US disclosed