SCHEMBL10840293

SCHEMBL10840293

COc1ccc(N([C]=O)Cc2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
LMNA P02545 2/20 0.50
NR3C1 P04150 1/20 0.50
PGR P06401 1/20 0.50
RNF4 P78317 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
ACHE P22303 1/20 0.49
LTA4H P09960 1/20 0.49
CNR1 P21554 2/20 0.48
CNR2 P34972 2/20 0.48
MAPK1 P28482 1/20 0.48
TSHR P16473 1/20 0.48
G6PC1 P35575 1/20 0.47
TRPM8 Q7Z2W7 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
TAS2R14 Q9NYV8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL305633 0.82 TSHR (0.45) ALDH1A1LMNATSHRTRPM8
SCHEMBL2093212 0.81 CYP2C19 (0.59) ALDH1A1LMNANR3C1NPSR1CNR1
SCHEMBL5541684 0.80 TP53 (0.48) ALDH1A1LMNACNR1CNR2TSHR
SCHEMBL2085584 0.78 KCNA5 (0.44) NR3C1CNR1CNR2TDP1TAS2R14
SCHEMBL2096014 0.78 HTR2A (0.40) ALDH1A1CNR2TSHR
SCHEMBL2094147 0.78 CNR1 (0.43) NR3C1PGRCNR1CNR2G6PC1
SCHEMBL2091209 0.78 L3MBTL1 (0.43) ALDH1A1LMNANR3C1CNR2MAPK1
SCHEMBL27787417 0.78 MAOB (0.44) ALDH1A1NR3C1CNR2TSHRTDP1
SCHEMBL7001778 0.78 CYP2C19 (0.63) ALDH1A1LMNANR3C1PGRRNF4
SCHEMBL5544762 0.77 NR1H4 (0.48) ALDH1A1LMNAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4617401-A ANTISPASMODIC AGENTS, VASODILATORS SUNTORY LTD. (JP) 1986-10-14 US claimed
EP-0039903-A2 8-Substituted pyrrolizidines and quaternary ammonium salts thereof SUNTORY KABUSHIKI KAISHA (JP) 1981-11-18 EP claimed
US-4617401-A ANTISPASMODIC AGENTS, VASODILATORS SUNTORY LTD. (JP) 1986-10-14 US disclosed
EP-0039903-A2 8-Substituted pyrrolizidines and quaternary ammonium salts thereof SUNTORY KABUSHIKI KAISHA (JP) 1981-11-18 EP disclosed