SCHEMBL10854890

SCHEMBL10854890

COc1ccc(C=C2CCn3c2nc2cc(NC(=O)CC(=O)O)ccc2c3=O)cc1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NME2 P22392 2/20 0.60
KMT2A Q03164 5/20 0.56
MEN1 O00255 4/20 0.56
MAPT P10636 2/20 0.56
RAB9A P51151 2/20 0.56
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 2/20 0.56
MCL1 Q07820 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
POLB P06746 1/20 0.55
THRB P10828 1/20 0.55
HPGD P15428 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
NPC1 O15118 1/20 0.53
CCR3 P51677 1/20 0.52
ALOX5 P09917 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10854883 1.00 NME2 (0.60) NME2KMT2AMEN1MAPTRAB9A
SCHEMBL10858565 0.93 NME2 (0.62) NME2KMT2AMEN1MAPTRAB9A
SCHEMBL10858584 0.93 NME2 (0.62) NME2KMT2AMEN1MAPTRAB9A
SCHEMBL10853231 0.92 KMT2A (0.59) NME2KMT2AMEN1MAPTRAB9A
SCHEMBL10853242 0.92 KMT2A (0.59) NME2KMT2AMEN1MAPTRAB9A
SCHEMBL10858499 0.91 NME2 (0.63) NME2KMT2AMEN1MAPTRAB9A
SCHEMBL10858502 0.91 NME2 (0.63) NME2KMT2AMEN1MAPTRAB9A
SCHEMBL10857243 0.91 NME2 (0.55) NME2KMT2AMEN1MAPTRAB9A
SCHEMBL10857248 0.91 NME2 (0.55) NME2KMT2AMEN1MAPTRAB9A
SCHEMBL10854992 0.90 KMT2A (0.58) NME2KMT2AMEN1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4579847-A Amino derivatives of benzylidene-pyrrolo[2,1-b]quinazolines useful for treating conditions of allergic origin FARMITALIA CARLO ERBA S.P.A. (IT) 1986-04-01 US disclosed