SCHEMBL10857643

SCHEMBL10857643

C=CC1(O)CCCc2c(OC)cccc21

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
CYP3A4 P08684 2/20 0.42
MAPT P10636 1/20 0.40
SIGMAR1 Q99720 1/20 0.39
SRD5A1 P18405 3/20 0.38
SRD5A2 P31213 3/20 0.38
PARP1 P09874 1/20 0.36
KMT2A Q03164 1/20 0.35
NOTUM Q6P988 1/20 0.34
PDK2 Q15119 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
HSD11B1 P28845 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11027320 0.82 PARP1 (0.41) ALDH1A1CYP3A4MAPTPARP1KMT2A
SCHEMBL13167579 0.79 ALDH1A1 (0.49) ALDH1A1CYP3A4MAPTSIGMAR1SRD5A1
SCHEMBL13185549 0.75 ALDH1A1 (0.43) ALDH1A1CYP3A4MAPTSIGMAR1SRD5A1
SCHEMBL12260114 0.75 ALDH1A1 (0.51) ALDH1A1CYP3A4MAPTSIGMAR1SRD5A1
SCHEMBL17014495 0.75 ALDH1A1 (0.48) ALDH1A1CYP3A4MAPTSIGMAR1SRD5A1
SCHEMBL7958551 0.74 ALDH1A1 (0.42) ALDH1A1CYP3A4MAPTSIGMAR1SRD5A1
SCHEMBL7565934 0.74 ALDH1A1 (0.42) ALDH1A1CYP3A4MAPTSIGMAR1SRD5A1
SCHEMBL6582087 0.74 ALDH1A1 (0.48) ALDH1A1CYP3A4MAPTSIGMAR1SRD5A1
SCHEMBL8139004 0.74 ALDH1A1 (0.44) ALDH1A1CYP3A4MAPTSIGMAR1SRD5A1
SCHEMBL7968392 0.73 ALDH1A1 (0.47) ALDH1A1CYP3A4MAPTSIGMAR1SRD5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4590274-A Antihypertensive 1-[bis-(substituted phenyl)methyl]-4[2-(1,2,3,4-tetrahydro-substituted naphthalen-1-ylidene)ethyl]piperazines E. I. DU PONT DE NEMOURS AND COMPANY (US) 1986-05-20 US disclosed