Stallimycin

Stallimycin

SCHEMBL108585

Cn1cc(NC(=O)c2cc(NC(=O)c3cc(NC=O)cn3C)cn2C)cc1C(=O)NCCC(=N)N

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRAS P01112 14/20 1.00
ESR1 P03372 13/20 1.00
ESR2 Q92731 13/20 1.00
TOP1 P11387 2/20 1.00
KDM4E B2RXH2 1/20 0.98
POLB P06746 1/20 0.98
MAPT P10636 1/20 0.98
HIF1A Q16665 1/20 0.98
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HPSE Q9Y251 1/20 0.34
P2RY12 Q9H244 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14002814 1.00 HRAS (1.00) HRASESR1ESR2TOP1KDM4E
Stallimycin SCHEMBL193003 0.99 KDM4E (1.00) HRASESR1ESR2TOP1KDM4E
SCHEMBL7125320 0.91 HRAS (0.83) HRASESR1ESR2TOP1KDM4E
SCHEMBL9714123 0.90 HRAS (0.81) HRASESR1ESR2TOP1KDM4E
SCHEMBL22590340 0.89 HRAS (0.80) HRASESR1ESR2TOP1KDM4E
Hydrochloric Acid SCHEMBL29375648 0.89 KDM4E (0.82) HRASESR1ESR2TOP1KDM4E
SCHEMBL30469493 0.88 HRAS (0.79) HRASESR1ESR2TOP1KDM4E
SCHEMBL29394871 0.87 HRAS (0.78) HRASESR1ESR2TOP1KDM4E
SCHEMBL6499316 0.87 HRAS (0.77) HRASESR1ESR2TOP1KDM4E
SCHEMBL7123738 0.87 HRAS (0.77) HRASESR1ESR2TOP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2086 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4667572-A2 THERAPEUTIC TREATMENT OF MICROSATELLITE UNSTABLE CANCERS The Broad Institute Inc. (US) 2025-12-24 EP claimed
EP-3802557-B1 THERAPEUTIC TREATMENT OF MICROSATELLITE UNSTABLE CANCERS BROAD INST INC (US) 2025-08-06 EP claimed
US-12337065-B2 Compositions for treating viral infections and methods for same ACCESS TO ADVANCED HEALTH INSTITUTE (US) 2025-06-24 US claimed
US-20250193430-A1 MULTIPLE TRANSFORMS ADJUSTMENT STAGES FOR VIDEO CODING QUALCOMM INCORPORATED 2025-06-12 US claimed
WO-2025059144-A1 DYNAMIC NANOMECHANICAL AMPLIFICATION ANTENNA AND USES SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2025-03-20 WO claimed
US-12256092-B2 Multiple transforms adjustment stages for video coding QUALCOMM INCORPORATED (US) 2025-03-18 US claimed
US-12246004-B2 Therapeutic treatment of microsatellite unstable cancers THE BROAD INSTITUTE, INC. (US) 2025-03-11 US claimed
US-20240417785-A1 ENHANCEMENT OF NUCLEIC ACID POLYMERIZATION BY MINOR GROOVE BINDING MOIETIES ROCHE SEQUENCING SOLUTIONS INC (US) 2024-12-19 US claimed
EP-3735477-B1 ENHANCEMENT OF NUCLEIC ACID POLYMERIZATION BY MINOR GROOVE BINDING MOIETIES ROCHE DIAGNOSTICS GMBH (DE) 2024-10-30 EP claimed
CN-118697017-A Sweetness and taste improvement of steviol glycoside or mogroside sweetener with flavonoids 可口可乐公司 2024-09-27 CN claimed
EP-0316440-B1 System and method for providing localized Mössbauer absorption in an organic medium MILLS RANDELL L (US) 1996-01-03 EP claimed
EP-0599188-A1 Trans and CIS traumatic acid salts having cicatrizant activity associated to bacteriostatic, antiviral, antibiotic or antifungal activity LIFEGROUP S.p.A. (IT) 1994-06-01 EP claimed
EP-0388948-B1 Acryloyl substituted pyrrole derivatives ERBA CARLO SPA (IT) 1993-12-15 EP claimed
EP-0246868-B1 SITE SPECIFIC ALKYLATING AGENTS FARMITALIA CARLO ERBA S.r.l. (IT) 1992-09-16 EP claimed
WO-1992009574-A2 POLY-AMINOPYRROLECARBOXAMIDO DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1992-06-11 WO claimed
EP-0450594-A2 DNA probe signal amplification Segev, David (US) 1991-10-09 EP claimed
EP-0416075-A1 ACRYLOYL SUBSTITUTED PYRROLE DERIVATIVES FARMITALIA CARLO ERBA S.r.l. (IT) 1991-03-13 EP claimed
WO-1990011277-A1 ACRYLOYL SUBSTITUTED PYRROLE DERIVATIVES FARMITALIA CARLO ERBA S.R.L. (IT) 1990-10-04 WO claimed
EP-0388948-A1 Acryloyl substituted pyrrole derivatives FARMITALIA CARLO ERBA S.r.l. (IT) 1990-09-26 EP claimed
EP-0246868-A1 Site specific alkylating agents FARMITALIA CARLO ERBA S.r.l. (IT) 1987-11-25 EP claimed