4-Hydroxy-Alprazolam

4-Hydroxy-Alprazolam

SCHEMBL10891720

Cc1nnc2n1-c1ccc(Cl)cc1C(c1ccccc1)=NC2O

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 14/20 0.60
BRD2 P25440 5/20 0.60
BRD3 Q15059 4/20 0.60
OPRK1 P41145 4/20 0.60
LMNA P02545 3/20 0.60
PDE3A Q14432 1/20 0.60
GABRA1 P14867 3/20 0.58
GABRA5 P31644 3/20 0.58
GABRA3 P34903 3/20 0.58
GABRA2 P47869 3/20 0.58
GABRB2 P47870 2/20 0.58
HPGD P15428 1/20 0.58
CNR1 P21554 1/20 0.58
CCKBR P32239 1/20 0.55
MEN1 O00255 1/20 0.47
ALB P02768 1/20 0.47
KMT2A Q03164 1/20 0.47
ADRA1A P35348 2/20 0.47
PDE4D Q08499 2/20 0.47
GABRG2 P18507 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
4-Hydroxy-Alprazolam SCHEMBL30150892 1.00 BRD4 (0.60) BRD4BRD2BRD3OPRK1LMNA
4-Hydroxy-Alprazolam SCHEMBL30150893 1.00 BRD4 (0.60) BRD4BRD2BRD3OPRK1LMNA
4-Hydroxy-Alprazolam SCHEMBL10890275 0.94 BRD4 (0.60) BRD4BRD2BRD3OPRK1LMNA
SCHEMBL11390416 0.86 BRD4 (0.58) BRD4BRD2BRD3OPRK1LMNA
SCHEMBL7903000 0.85 BRD4 (0.62) BRD4BRD2BRD3OPRK1LMNA
SCHEMBL7895743 0.85 BRD4 (0.60) BRD4BRD2BRD3OPRK1LMNA
SCHEMBL11901048 0.84 BRD4 (0.77) BRD4BRD2BRD3OPRK1LMNA
SCHEMBL7903005 0.83 BRD4 (0.75) BRD4BRD2BRD3LMNASLC6A3
SCHEMBL11828757 0.83 OPRK1 (0.58) BRD4BRD2BRD3OPRK1LMNA
SCHEMBL11705304 0.82 BRD4 (0.61) BRD4BRD2BRD3OPRK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4588721-A Treatment of negative symptoms of schizophrenia THE UPJOHN COMPANY (US) 1986-05-13 US claimed
EP-0139460-A2 Benzodiazepines and their therapeutic use THE UPJOHN COMPANY (US) 1985-05-02 EP claimed
US-4044016-A ANTICONVULSANTS, SEDATIVES, MUSCLE RELAXANTS HOFFMANN-LA ROCHE INC. (US) 1977-08-23 US disclosed
US-3970664-A ANTICONVULSANT, MUSCLE RELAXANT, SEDATIVE HOFFMANN-LA ROCHE INC. (US) 1976-07-20 US disclosed
US-3954728-A ANTICONVULSANTS, MUSCLE RELAXANTS, SEDATIVES HOFFMAN-LA ROCHE INC. (US) 1976-05-04 US disclosed