SCHEMBL10897269

SCHEMBL10897269

COc1cc2onc(C3CCNCC3)c2cc1OC

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.43
JUND P17535 1/20 0.42
FOSB P53539 1/20 0.42
HTR2C P28335 3/20 0.41
TLR9 Q9NR96 2/20 0.39
TLR7 Q9NYK1 2/20 0.39
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
TLR8 Q9NR97 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL10637114 0.99 MAPK14 (0.43) MAPK14JUNDFOSBHTR2CTLR9
SCHEMBL11236323 0.81 HTR2C (0.47) MAPK14JUNDFOSBHTR2CDRD2
SCHEMBL10897405 0.81 MAPK14 (0.47) MAPK14JUNDFOSBHTR2CDRD2
Bromide SCHEMBL10641053 0.80 MAPK14 (0.46) MAPK14JUNDFOSBHTR2CDRD2
Hydrochloric Acid SCHEMBL29688457 0.80 HTR2C (0.48) MAPK14JUNDFOSBHTR2CDRD2
Hydrochloric Acid SCHEMBL1833385 0.80 HTR2C (0.48) MAPK14JUNDFOSBHTR2CDRD2
SCHEMBL1838388 0.77 QDPR (0.48) HTR2CDRD2HTR2A
SCHEMBL23595431 0.76 HTR2A (0.48) MAPK14TLR9TLR7DRD2HTR2A
SCHEMBL14034032 0.75 HTR2A (0.46) MAPK14HTR2CDRD2HTR2A
SCHEMBL470707 0.75 MAPK14 (0.52) MAPK14HTR2CDRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4355037-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS (US) 1982-10-19 US claimed
EP-0079564-B1 3-(1-SUBSTITUTED-4-PIPERIDYL)-1,2-BENZISOXAZOLES, A PROCESS FOR THE PREPARATION THEREOF, A PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1986-03-19 EP disclosed
EP-0079564-A1 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles, a process for the preparation thereof, a pharmaceutical composition comprising the same, and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1983-05-25 EP disclosed
US-4352811-A NEUROLEPTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1982-10-05 US disclosed