SCHEMBL10899211

SCHEMBL10899211

CC(C)(C)OC(=O)CNn1cc(C(=O)O)c(=O)c2cc(F)c(F)c(F)c21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.43
ALDH1A1 P00352 6/20 0.43
POLB P06746 1/20 0.43
HSP90AA1 P07900 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
TOP2A P11388 3/20 0.38
TOP2B Q02880 3/20 0.38
STAT3 P40763 2/20 0.38
TOP1 P11387 1/20 0.37
HPGD P15428 4/20 0.37
HSD17B10 Q99714 3/20 0.37
PMP22 Q01453 1/20 0.36
DRD3 P35462 1/20 0.36
BRD4 O60885 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
CYP2J2 P51589 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KMT2A Q03164 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2023894 0.79 KDM4E (0.48) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL3290754 0.76 KMT2A (0.42) KDM4EALDH1A1STAT3HPGDHSD17B10
SCHEMBL10899205 0.75 KDM4E (0.44) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL13326853 0.74 STAT3 (0.52) KDM4EALDH1A1STAT3HPGDHSD17B10
SCHEMBL8136260 0.74 TOP2A (0.53) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL10654436 0.72 KDM4E (0.51) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL10901383 0.72 KDM4E (0.41) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL500816 0.71 KDM4E (0.61) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL30843076 0.71 KDM4E (0.61) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL9572075 0.71 STAT3 (0.56) KDM4EALDH1A1STAT3HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4604401-A QUINOLINE-CARBOXYLIC ACIDS WARNER-LAMBERT COMPANY (US) 1986-08-05 US disclosed
EP-0169710-A2 7-Substituted-6-fluoro-8-substituted-1,4-dihydro-1-methylamino-4-oxo-3-quinolinecarboxylic acids; 7-substituted-6-fluoro-1,4-dihydro-1-methylamino-4-oxo-3-naphthyridine carboxylic acids; derivatives thereof; and processes for producing the compounds WARNER-LAMBERT COMPANY (US) 1986-01-29 EP disclosed