SCHEMBL10899205

SCHEMBL10899205

CN(C(=O)OC(C)(C)C)n1cc(C(=O)O)c(=O)c2cc(F)c(F)c(F)c21

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.44
ALDH1A1 P00352 5/20 0.44
POLB P06746 1/20 0.44
HSP90AA1 P07900 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
TOP1 P11387 1/20 0.37
TOP2A P11388 5/20 0.37
TOP2B Q02880 5/20 0.37
STAT3 P40763 1/20 0.37
HPGD P15428 3/20 0.35
HSD17B10 Q99714 3/20 0.35
ADRA2B P18089 1/20 0.35
MAPK1 P28482 1/20 0.35
PMP22 Q01453 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
CYP1A2 P05177 1/20 0.34
DRD3 P35462 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9427167 0.90 STAT3 (0.38) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL9427196 0.87 STAT3 (0.52) KDM4EALDH1A1STAT3HPGDHSD17B10
SCHEMBL6213034 0.82 KDM4E (0.48) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL9289491 0.78 KDM4E (0.45) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL13326854 0.76 STAT3 (0.48) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL10899211 0.75 KDM4E (0.43) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL8136260 0.74 TOP2A (0.53) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL3290751 0.74 STAT3 (0.41) KDM4EALDH1A1STAT3HPGDHSD17B10
SCHEMBL10654436 0.73 KDM4E (0.51) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL25335713 0.72 LMNA (0.30) HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4604401-A QUINOLINE-CARBOXYLIC ACIDS WARNER-LAMBERT COMPANY (US) 1986-08-05 US disclosed
EP-0169710-A2 7-Substituted-6-fluoro-8-substituted-1,4-dihydro-1-methylamino-4-oxo-3-quinolinecarboxylic acids; 7-substituted-6-fluoro-1,4-dihydro-1-methylamino-4-oxo-3-naphthyridine carboxylic acids; derivatives thereof; and processes for producing the compounds WARNER-LAMBERT COMPANY (US) 1986-01-29 EP disclosed