SCHEMBL10900596

SCHEMBL10900596

COC(C(N)=O)C(=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.45
MAPT P10636 4/20 0.45
TDP1 Q9NUW8 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
CYP3A4 P08684 2/20 0.45
POLB P06746 2/20 0.45
PARP1 P09874 1/20 0.45
CYP2C19 P33261 1/20 0.45
RECQL P46063 1/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
HSD17B10 Q99714 1/20 0.45
ALDH1A1 P00352 3/20 0.43
LMNA P02545 3/20 0.42
CES2 O00748 2/20 0.42
CES1 P23141 2/20 0.42
HTT P42858 2/20 0.41
PGR P06401 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL146504 0.88 TSHR (0.52) TSHRMAPTTDP1L3MBTL1CYP3A4
SCHEMBL27285922 0.84 TSHR (0.48) TSHRMAPTTDP1L3MBTL1CYP3A4
SCHEMBL8665164 0.82 ALDH1A1 (0.49) TSHRMAPTTDP1L3MBTL1CYP3A4
SCHEMBL28783553 0.82 ALDH1A1 (0.49) TSHRMAPTTDP1L3MBTL1CYP3A4
SCHEMBL22209161 0.79 TDP1 (0.43) TSHRMAPTTDP1L3MBTL1CYP3A4
SCHEMBL28683232 0.77 KMT2A (0.54) TSHRMAPTTDP1POLBALDH1A1
SCHEMBL4644411 0.77 KMT2A (0.54) TSHRMAPTTDP1POLBALDH1A1
SCHEMBL1932808 0.77 CES1 (0.46) TSHRMAPTTDP1L3MBTL1CYP3A4
SCHEMBL10772180 0.77 AKR1C3 (0.48) TSHRMAPTTDP1L3MBTL1CYP3A4
SCHEMBL2231539 0.76 TSHR (0.48) TSHRMAPTTDP1L3MBTL1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019008154-A1 3-(AZOLYLMETHOXY)BIPHENYL DERIVATIVES AS INHIBITORS OF THE PD-1/PD-L1 PROTEIN/PROTEIN INTERACTION RIJKSUNIVERSITEIT GRONINGEN (NL) 2019-01-10 WO disclosed
CN-1088709-C Amine compound and its acid addition salt ROUSSEL UCLAF (FR) 2002-08-07 CN disclosed
CN-1052984-C Novel erythromycin derivatives, process for their preparation and their use as medicaments ROUSSEL UCLAF (FR) 2000-05-31 CN disclosed
CN-1229082-A Amine compound and its acid addition salt ROUSSEL UCLAF (FR) 1999-09-22 CN disclosed
CN-1151746-A Novel erythromycin derivatives, process for their preparation and their use as medicaments ROUSSEL UCLAF (FR) 1997-06-11 CN disclosed
EP-0087237-B1 CARBACYCLIN ANALOGUES THE UPJOHN COMPANY (US) 1986-05-14 EP disclosed