SCHEMBL1090665

SCHEMBL1090665

CC(C)c1ccc(Cl)nc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.44
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
SLC6A2 P23975 3/20 0.41
SLC6A4 P31645 3/20 0.41
SLC6A3 Q01959 3/20 0.41
KCNH2 Q12809 1/20 0.41
PIK3CD O00329 1/20 0.39
NAPRT Q6XQN6 1/20 0.39
NFKB1 P19838 1/20 0.38
TYR P14679 1/20 0.38
LMNA P02545 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15643867 0.84 SMN1; SMN2 (0.43) SMN1; SMN2CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL4252351 0.84 SMN1; SMN2 (0.43) SMN1; SMN2CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL1856238 0.84 SMN1; SMN2 (0.43) SMN1; SMN2CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL594060 0.82 CYP3A4 (0.42) SMN1; SMN2CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL21202536 0.82 SMN1; SMN2 (0.42) SMN1; SMN2CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL14358057 0.82 SMN1; SMN2 (0.42) SMN1; SMN2CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL17000183 0.82 SMN1; SMN2 (0.42) SMN1; SMN2CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL4092765 0.82 ADRB2 (0.52) SMN1; SMN2CYP3A4CYP2D6SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL8572234 0.82 SMN1; SMN2 (0.42) SMN1; SMN2CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL14127344 0.82 SMN1; SMN2 (0.42) SMN1; SMN2CYP3A4CYP2D6SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 535 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0897914-B1 Process for the preparation of 2,5-disubstitued pyridines HOFFMANN LA ROCHE (CH) 2004-05-26 EP claimed
US-6080866-A A CHEMICAL INTERMEDIATES FOR ENDOTHELIN RECEPTOR ANTAGONISTS HOFFMANN-LA ROCHE INC. (US) 2000-06-27 US claimed
CN-1210105-A Process for preparation of 2,5-disubstituted pyridines HOFFMANN LA ROCHE (CH) 1999-03-10 CN claimed
EP-0897914-A1 Process for the preparation of 2,5-disubstitued pyridines F. HOFFMANN-LA ROCHE AG (CH) 1999-02-24 EP claimed
JP-11116554-A None JP disclosed
EP-4448492-B1 COMPOSITIONS AND METHODS OF MAKING AND USING SMALL MOLECULES IN THE TREATMENT OF CANCER REGLAGENE INC (US) 2026-03-04 EP disclosed
WO-2025245178-A1 PAK4, CSTF2, OR CSTF2T PROTEIN DEGRADERS, PHARMACEUTICAL COMPOSITIONS, AND THERAPEUTIC APPLICATIONS INNOVO THERAPEUTICS, INC. (US) 2025-11-27 WO disclosed
US-12404242-B2 Compositions and methods for making and using small molecules in the treatment of cancer REGLAGENE, INC. (US) 2025-09-02 US disclosed
US-20250163063-A1 INHIBITORS OF CDK4/6 KINASE KHORA SPV 1, LLC 2025-05-22 US disclosed
US-20250109105-A1 COMPOSITIONS AND METHODS FOR MAKING AND USING SMALL MOLECULES IN THE TREATMENT OF CANCER REGLAGENE, INC. 2025-04-03 US disclosed
EP-4081523-B1 SUBSTITUTED BICYCLIC PIPERIDINE DERIVATIVES USEFUL AS T CELL ACTIVATORS BRISTOL MYERS SQUIBB CO (US) 2024-12-25 EP disclosed
EP-4469062-A1 INHIBITORS OF CDK4/6 KINASE Kinnate Biopharma Inc. (US) 2024-12-04 EP disclosed
EP-1483265-A1 PURINE DERIVATIVES AS KINASE INHIBITORS ELI LILLY AND COMPANY (US) 2004-12-08 EP disclosed
EP-0897914-B1 Process for the preparation of 2,5-disubstitued pyridines HOFFMANN LA ROCHE (CH) 2004-05-26 EP disclosed
WO-2003076442-A1 PURINE DERIVATIVES AS KINASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-09-18 WO disclosed
CN-1103335-C Process for preparation of 2,5-disubstituted pyridines HOFFMANN LA ROCHE (CH) 2003-03-19 CN disclosed
US-6080866-A A CHEMICAL INTERMEDIATES FOR ENDOTHELIN RECEPTOR ANTAGONISTS HOFFMANN-LA ROCHE INC. (US) 2000-06-27 US disclosed
CN-1210105-A Process for preparation of 2,5-disubstituted pyridines HOFFMANN LA ROCHE (CH) 1999-03-10 CN disclosed
EP-0897914-A1 Process for the preparation of 2,5-disubstitued pyridines F. HOFFMANN-LA ROCHE AG (CH) 1999-02-24 EP disclosed
US-4348396-A Substituted 11-oxo-11H-pyrido[2,1-b]quinazolines and method of inhibiting allergic reactions with them HOFFMANN-LA ROCHE INC. (US) 1982-09-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250109105-A1 COMPOSITIONS AND METHODS FOR MAKING AND USING SMALL MOLECULES IN THE TREATMENT OF CANCER CD47, RB1, TP53 SMN1; SMN2 159/4885CYP3A4 4626/4885CYP2D6 2951/4885
US-20250163063-A1 INHIBITORS OF CDK4/6 KINASE CDK4, CDK6, CDK2 SMN1; SMN2 2089/4885CYP3A4 3804/4885CYP2D6 2098/4885
US-12404242-B2 Compositions and methods for making and using small molecules in the treatment of cancer CD47, RB1, TP53 SMN1; SMN2 159/4885CYP3A4 4626/4885CYP2D6 2951/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.