SCHEMBL10909031

SCHEMBL10909031

NCCCNCc1cccc(Cl)c1

nearest known ligand 0.77

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.77
MC4R P32245 2/20 0.57
MC5R P33032 2/20 0.57
MC3R P41968 1/20 0.57
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C19 P33261 1/20 0.55
ACHE P22303 4/20 0.55
TAAR1 Q96RJ0 1/20 0.55
PNMT P11086 2/20 0.53
MAOA P21397 1/20 0.48
FOLH1 Q04609 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9903568 0.93 CHRM2 (0.77) CHRM2MC4RMC5RCYP1A2CYP3A4
SCHEMBL11673587 0.89 CHRM2 (0.89) CHRM2CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL16151774 0.87 MC4R (0.66) CHRM2MC4RMC5RMC3RCYP1A2
SCHEMBL7774786 0.85 CHRM2 (0.81) CHRM2CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL16260100 0.84 CHRM2 (0.62) CHRM2MC4RMC5RMC3RCYP1A2
SCHEMBL16136721 0.84 MC4R (0.62) CHRM2MC4RMC5RMC3RCYP1A2
SCHEMBL16152234 0.84 MC4R (0.62) CHRM2MC4RMC5RMC3RCYP1A2
SCHEMBL16152208 0.84 CHRM2 (0.62) CHRM2MC4RMC5RMC3RCYP1A2
SCHEMBL17770844 0.84 CHRM2 (0.62) CHRM2MC4RMC5RMC3RCYP1A2
SCHEMBL13975775 0.83 CHRM2 (0.77) CHRM2CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007117180-A1 AZAHETEROCYCLES, COMBINATORY LIBRARY, FOCUSED LIBRARY, PHARMACEUTICAL COMPOSITION AND METHODS FOR THE PRODUCTION THEREOF 'CHEMICAL DIVERSITY RESEARCH INSTITUTE' LTD. (RU) 2007-10-18 WO disclosed
US-4590272-A INSECTICIDES, MITICIDES, NEMATOCIDES NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1986-05-20 US disclosed
EP-0136636-A2 Nitromethylene-tetrahydropyrimidine derivatives, process for their preparation and insecticidal, miticidal, tickicidal, and nematicidal means NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1985-04-10 EP disclosed