SCHEMBL10944003

SCHEMBL10944003

OC[C@H]1O[C@@H](n2cnc3c(NC4Cc5ccccc5C4)ncnc32)[C@H](O)[C@@H]1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.75
PMP22 Q01453 2/20 0.75
ADORA2A P29274 2/20 0.75
ADORA3 P0DMS8 1/20 0.75
GAA P10253 1/20 0.75
ADORA2B P29275 1/20 0.75
ADORA1 P30542 1/20 0.75
HTT P42858 1/20 0.75
SIGMAR1 Q99720 1/20 0.75
SLC29A1 Q99808 1/20 0.75
RXFP1 Q9HBX9 1/20 0.75
MEN1 O00255 1/20 0.75
KMT2A Q03164 1/20 0.75
TP53 P04637 1/20 0.75
NFKB1 P19838 1/20 0.75
HIF1A Q16665 1/20 0.75
SMN1; SMN2 Q16637 1/20 0.74
TDP1 Q9NUW8 1/20 0.74
CYP2C19 P33261 1/20 0.74
THPO P40225 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11881650 0.94 TSHR (0.72) TSHRPMP22ADORA2AADORA3GAA
SCHEMBL9352957 0.89 MEN1 (0.76) TSHRPMP22ADORA2AADORA3GAA
SCHEMBL9352946 0.89 MEN1 (0.76) TSHRPMP22ADORA2AADORA3GAA
SCHEMBL23982261 0.88 ADORA1 (0.92) TSHRPMP22ADORA2AADORA3GAA
SCHEMBL9495163 0.88 ADORA1 (0.92) TSHRPMP22ADORA2AADORA3GAA
SCHEMBL9495177 0.88 ADORA1 (0.92) TSHRPMP22ADORA2AADORA3GAA
SCHEMBL9142235 0.88 ADORA1 (0.92) TSHRPMP22ADORA2AADORA3GAA
SCHEMBL11013427 0.86 TSHR (0.69) TSHRPMP22ADORA2AADORA3GAA
N6-Cyclopentyladenosine SCHEMBL472621 0.86 ADORA3 (1.00) TSHRPMP22ADORA2AADORA3GAA
SCHEMBL9793271 0.86 ADORA3 (0.96) TSHRPMP22ADORA2AADORA3GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4501735-A HYPOTENSIVE AGENTS WARNER-LAMBERT COMPANY (US) 1985-02-26 US disclosed