SCHEMBL10955871

SCHEMBL10955871

Cn1cnc2c1c(=O)n(Cc1ccc(C(C)(C)C)cc1)c(=O)n2C

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC8 Q09428 1/20 0.64
KCNJ11 Q14654 1/20 0.64
MAPK1 P28482 2/20 0.62
NPSR1 Q6W5P4 1/20 0.57
ADORA2B P29275 8/20 0.56
GLA P06280 1/20 0.55
BLM P54132 1/20 0.55
KMT2A Q03164 1/20 0.55
ACHE P22303 2/20 0.52
PIK3CD O00329 1/20 0.52
POLB P06746 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
CNR1 P21554 1/20 0.52
ADORA2A P29274 1/20 0.52
ADORA1 P30542 1/20 0.52
NTSR1 P30989 1/20 0.52
MC3R P41968 1/20 0.52
NOTUM Q6P988 1/20 0.52
SIRT3 Q9NTG7 1/20 0.52
GDA Q9Y2T3 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19601319 0.91 MAPK1 (0.58) ABCC8KCNJ11MAPK1NPSR1ADORA2B
SCHEMBL17682264 0.87 MAPK1 (0.54) ABCC8KCNJ11MAPK1NPSR1ADORA2B
SCHEMBL17682265 0.87 MAPK1 (0.56) ABCC8KCNJ11MAPK1NPSR1ADORA2B
SCHEMBL10394509 0.85 MAPK1 (0.73) MAPK1NPSR1ADORA2BGLABLM
Iodide SCHEMBL28480464 0.84 MAPK1 (0.72) MAPK1NPSR1ADORA2BGLABLM
SCHEMBL29148051 0.84 ADORA2B (0.62) MAPK1NPSR1ADORA2BGLABLM
SCHEMBL18989514 0.82 MAPK1 (0.66) MAPK1NPSR1ADORA2BGLABLM
SCHEMBL19601321 0.81 MAPK1 (0.55) MAPK1NPSR1ADORA2BGLABLM
SCHEMBL27699778 0.81 MAPK1 (0.67) MAPK1NPSR1ADORA2BGLABLM
SCHEMBL19601323 0.80 MAPK1 (0.69) MAPK1NPSR1ADORA2BGLABLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0019165-B1 PROCESS FOR PREPARING 1,3,7-TRIALKYLXANTHINES SOCIETE DES PRODUITS NESTLE S.A. (CH) 1985-07-31 EP disclosed
US-4450163-A ANTIBODY INHIBITORS; N-ALKYLATION OF XANTHINES USING PHASE TRANSFER AGENTS SOCIETE D'ASSISTANCE TECHNIQUE POUR PRODUITS NESTLE S.A. (CH) 1984-05-22 US disclosed
EP-0019165-A1 Process for preparing 1,3,7-trialkylxanthines SOCIETE DES PRODUITS NESTLE S.A. (CH) 1980-11-26 EP disclosed