SCHEMBL10959565

SCHEMBL10959565

C1=CC2(C=C3Sc4ccccc4N=C13)OO2

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.32
TRPA1 O75762 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28807038 0.83 BACE1 (0.33) BACE1TRPA1
SCHEMBL27930103 0.81 BACE1 (0.35) BACE1TRPA1
SCHEMBL27662416 0.81 BACE1 (0.35) BACE1TRPA1
SCHEMBL28001724 0.79 BACE1 (0.31) BACE1
SCHEMBL27930647 0.79 BACE1 (0.31) BACE1
SCHEMBL28206346 0.79 BACE1 (0.31) BACE1
SCHEMBL27423963 0.78 BACE1 (0.30) BACE1
SCHEMBL28110668 0.78 BACE1 (0.30) BACE1
SCHEMBL27548732 0.72 MMP2 (0.31)
SCHEMBL28461077 0.71 BACE1 (0.33) BACE1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0136893-A2 Benzo[a]phenothiazines and hydro-derivatives and pharmaceutical compositions containing them MERCK FROSST CANADA INC. (CA) 1985-04-10 EP claimed