SCHEMBL10965335

SCHEMBL10965335

Cc1[nH]c(=O)c(C(N)=O)cc1-c1csc(-c2cccnc2)n1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 5/20 0.56
CDK5R1 Q15078 5/20 0.56
CYP17A1 P05093 1/20 0.53
CYP19A1 P11511 5/20 0.52
AXL P30530 1/20 0.52
PBRM1 Q86U86 1/20 0.52
MKNK1 Q9BUB5 1/20 0.52
MKNK2 Q9HBH9 1/20 0.52
RAB9A P51151 5/20 0.51
NPC1 O15118 4/20 0.51
MAPT P10636 2/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
TDP1 Q9NUW8 2/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10966927 0.88 CDK5 (0.64) CDK5CDK5R1MEN1KMT2A
SCHEMBL11078693 0.84 MKNK1 (0.56) MKNK1MKNK2KMT2A
SCHEMBL10965295 0.84 MEN1 (0.52) CDK5CDK5R1RAB9ANPC1MEN1
SCHEMBL10965672 0.83 CDK5 (0.54) CDK5CDK5R1CYP19A1RAB9AMAPT
SCHEMBL10964379 0.83 CDK5 (0.54) CDK5CDK5R1RAB9ANPC1MEN1
SCHEMBL10966867 0.82 CDK5 (0.52) CDK5CDK5R1RAB9ANPC1MEN1
SCHEMBL10966720 0.82 MEN1 (0.50) CDK5CDK5R1RAB9ANPC1MEN1
SCHEMBL10965808 0.81 MEN1 (0.47) CDK5CDK5R1CYP19A1RAB9AMAPT
SCHEMBL10965193 0.81 HTR2B (0.50) CDK5CDK5R1CYP19A1RAB9ANPC1
SCHEMBL10963815 0.81 MAPT (0.51) CDK5CDK5R1RAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0154190-A1 Pyridones MERCK PATENT GmbH (DE) 1985-09-11 EP disclosed