SCHEMBL10967478

SCHEMBL10967478

CC(=O)Nc1ccc2ncnc(NC=C(C(=O)O)C(=O)O)c2c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.56
FYN P06241 6/20 0.49
SRC P12931 6/20 0.49
ABCG2 Q9UNQ0 1/20 0.49
VCP P55072 1/20 0.47
ERBB2 P04626 3/20 0.46
LCK P06239 1/20 0.46
MAP4K4 O95819 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11099669 0.90 EGFR (0.56) EGFRABCG2ERBB2MAP4K4
SCHEMBL10970610 0.87 FYN (0.48) EGFRFYNSRCVCPERBB2
SCHEMBL10966607 0.87 EGFR (0.48) EGFRFYNSRCVCPERBB2
SCHEMBL10967809 0.87 FYN (0.60) EGFRFYNSRCVCPERBB2
SCHEMBL10969619 0.86 FYN (0.53) EGFRFYNSRCERBB2
SCHEMBL10967974 0.85 FYN (0.47) EGFRFYNSRCVCPERBB2
SCHEMBL10971936 0.85 FYN (0.46) EGFRFYNSRCVCPERBB2
SCHEMBL10970261 0.85 FYN (0.52) EGFRFYNSRCVCPERBB2
SCHEMBL10967392 0.84 FYN (0.52) EGFRFYNSRCVCPERBB2
SCHEMBL10967279 0.84 EGFR (0.46) EGFRFYNSRCVCPERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4543356-A Quinazoline derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1985-09-24 US disclosed
EP-0030156-B1 QUINAZOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1984-03-21 EP disclosed
US-4429126-A ANTIASTHMA FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1984-01-31 US disclosed
US-4377580-A ANTIALLERGENIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-03-22 US disclosed
EP-0030156-A1 Quinazoline derivatives, processes for their preparation and pharmaceutical compositions containing them FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-06-10 EP disclosed