SCHEMBL10974166

SCHEMBL10974166

COc1ccc(-c2nc(CCl)nn2-c2ccc(OC)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.64
PTGS1 P23219 5/20 0.64
L3MBTL1 Q9Y468 1/20 0.49
MALT1 Q9UDY8 1/20 0.48
LMNA P02545 1/20 0.47
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MYOF Q9NZM1 1/20 0.43
GLA P06280 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13239884 0.90 PTGS1 (0.56) PTGS2PTGS1L3MBTL1MALT1CYP3A4
SCHEMBL10977699 0.85 PTGS2 (0.64) PTGS2PTGS1L3MBTL1MALT1LMNA
SCHEMBL10973892 0.82 PTGS2 (0.59) PTGS2PTGS1L3MBTL1MALT1LMNA
SCHEMBL13239881 0.81 PTGS1 (0.47) PTGS2PTGS1LMNACYP3A4CYP2C9
SCHEMBL10978842 0.81 PTGS2 (0.58) PTGS2PTGS1L3MBTL1MALT1LMNA
SCHEMBL13239896 0.80 PTGS1 (0.46) PTGS2PTGS1L3MBTL1MALT1LMNA
SCHEMBL1193845 0.78 PTGS2 (1.00) PTGS2PTGS1L3MBTL1MALT1LMNA
SCHEMBL6132166 0.77 PTGS2 (0.69) PTGS2PTGS1L3MBTL1MALT1LMNA
SCHEMBL3983431 0.77 PTGS2 (0.69) PTGS2PTGS1L3MBTL1LMNA
SCHEMBL4028727 0.77 PTGS2 (0.69) PTGS2PTGS1L3MBTL1MALT1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0162217-A1 1,2,4-Triazacycloalcadiene derivatives CIBA-GEIGY AG (CH) 1985-11-27 EP disclosed