SCHEMBL10977240

SCHEMBL10977240

Cc1nc(CC(=O)Nc2ccccc2)cs1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.71
TP53 P04637 2/20 0.71
SMN1; SMN2 Q16637 2/20 0.71
GAA P10253 2/20 0.71
MEN1 O00255 3/20 0.67
KMT2A Q03164 3/20 0.67
SLC12A2 P55011 1/20 0.67
SLC12A5 Q9H2X9 1/20 0.67
CYP1A2 P05177 1/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2D6 P10635 1/20 0.62
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
NPC1 O15118 1/20 0.61
RAB9A P51151 1/20 0.61
LMNA P02545 3/20 0.57
ALDH1A1 P00352 1/20 0.56
HPGD P15428 1/20 0.56
CTPS1 P17812 1/20 0.56
HTT P42858 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25720785 0.78 PDE5A (0.79) MAPTSMN1; SMN2MEN1KMT2ACYP1A2
SCHEMBL16770015 0.78 SMN1; SMN2 (0.57) MAPTTP53SMN1; SMN2GAAMEN1
Hydrochloric Acid SCHEMBL6622281 0.78 ADRB3 (0.80) MAPTTP53SMN1; SMN2GAA
Hydrochloric Acid SCHEMBL6622276 0.78 ADRB3 (0.80) MAPTTP53SMN1; SMN2GAA
SCHEMBL2409605 0.77 MEN1 (0.57) MAPTTP53SMN1; SMN2GAAMEN1
SCHEMBL1128988 0.76 SMN1; SMN2 (0.59) MAPTTP53SMN1; SMN2GAAMEN1
SCHEMBL26334694 0.76 SMN1; SMN2 (0.56) MAPTTP53SMN1; SMN2GAAMEN1
SCHEMBL23140029 0.76 CTPS1 (0.75) MAPTMEN1KMT2ASLC12A2SLC12A5
Hydrochloric Acid SCHEMBL826687 0.76 MEN1 (0.56) MAPTTP53SMN1; SMN2GAAMEN1
SCHEMBL5544118 0.76 MAPT (0.56) MAPTTP53SMN1; SMN2GAASLC12A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0066993-B1 QUINOLINE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-01-30 EP disclosed
US-4435405-A 2-(AMINOALKYLTHIO) SUBSTITUTED IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-03-06 US disclosed
EP-0066993-A1 Quinoline derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-12-15 EP disclosed