SCHEMBL10979593

SCHEMBL10979593

Oc1ccc(CN(O)Cc2ccc(O)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.54
ESR2 Q92731 3/20 0.54
ABAT P80404 1/20 0.48
CA2 P00918 4/20 0.46
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
BLM P54132 2/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
CA12 O43570 1/20 0.44
GMNN O75496 1/20 0.44
CA1 P00915 1/20 0.44
LMNA P02545 1/20 0.44
CA3 P07451 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
TYR P14679 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3804172 0.85 ALDH1A1 (0.52) ESR1ESR2ABATCA2ALDH1A1
SCHEMBL29369685 0.80 ESR1 (0.55) ESR1ESR2ABATCA2ALDH1A1
SCHEMBL22477359 0.79 ESR1 (0.48) ESR1ESR2ABATCA2ALDH1A1
SCHEMBL15490714 0.79 ESR1 (0.80) ESR1ESR2ABATCA2ALDH1A1
SCHEMBL10748300 0.78 CYP1A2 (0.53) CA2ALDH1A1NPC1CA12CA1
SCHEMBL8781904 0.78 TSHR (0.46) ESR1ESR2CA2CA12CA1
SCHEMBL116611 0.76 HRH3 (0.64) ESR1ESR2ABATCA2ALDH1A1
SCHEMBL9416592 0.76 BCHE (0.53) ESR1ESR2ABATCA2ALDH1A1
SCHEMBL19206134 0.76 HRH3 (0.64) ESR1ESR2ABATCA2ALDH1A1
SCHEMBL4967718 0.76 CYP2C19 (0.50) ALDH1A1IDO1TAAR1CYP2C19TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112190570-B Application of gastrodia tuber source derivative in preparing medicine for treating acute or chronic pain 中国医学科学院药物研究所 2023-05-05 CN disclosed
CN-112190571-B Application of gastrodia tuber source derivative in preparing medicine for treating inflammatory bowel disease 中国医学科学院药物研究所 2023-05-05 CN disclosed
CN-112190571-A Application of derivative from gastrodia elata in preparation of medicine for treating inflammatory bowel disease 中国医学科学院药物研究所 2021-01-08 CN disclosed
CN-112190570-A Application of derivative derived from rhizoma gastrodiae in preparation of medicine for treating acute or chronic pain 中国医学科学院药物研究所 2021-01-08 CN disclosed
CN-103420805-B Polybenzyl derivatives with nerve cell protective activity in tall gastrodia tuber 中国医学科学院药物研究所 2017-04-26 CN disclosed
CN-103420805-A Polybenzyl derivatives with nerve cell protective activity in tall gastrodia tuber INST MATERIA MEDICA CAMS 2013-12-04 CN disclosed
EP-0140378-A2 Discoloration-resistant spandex fiber E.I. DU PONT DE NEMOURS AND COMPANY (US) 1985-05-08 EP disclosed