SCHEMBL10984029

SCHEMBL10984029

COc1ccc2cc(-c3nc4ncccc4[nH]3)ccc2c1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 7/20 0.80
PDE2A O00408 1/20 0.67
PRMT5 O14744 2/20 0.56
PDE5A O76074 2/20 0.54
FGFR1 P11362 1/20 0.54
FGFR2 P21802 1/20 0.54
FGFR3 P22607 1/20 0.54
NOS1 P29475 2/20 0.51
NOS2 P35228 2/20 0.51
CYP2C9 P11712 1/20 0.51
NPY5R Q15761 1/20 0.50
FAAH O00519 1/20 0.49
NOS3 P29474 1/20 0.49
TP53 P04637 1/20 0.49
HPSE Q9Y251 1/20 0.49
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
ALDH1A1 P00352 1/20 0.49
PKM P14618 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11772846 0.89 AURKA (1.00) AURKAPDE2APRMT5PDE5ATP53
SCHEMBL10981003 0.85 PDE2A (0.65) AURKAPDE2APRMT5PDE5AFGFR1
SCHEMBL7456059 0.84 AURKA (0.64) AURKAPRMT5PDE5ANPY5RFAAH
SCHEMBL10964336 0.80 AURKA (0.51) AURKAPDE2ACYP2C9NPY5RTP53
SCHEMBL11773596 0.80 PDE2A (0.81) AURKAPDE2APDE5AFGFR1FGFR2
SCHEMBL11770981 0.80 PDE2A (1.00) AURKAPDE2APDE5AKDM4EALDH1A1
SCHEMBL10983075 0.80 AURKA (0.64) AURKAPDE2APRMT5PDE5ANPY5R
Hydrochloric Acid SCHEMBL11769751 0.79 PDE2A (0.97) AURKAPDE2APDE5AKDM4EALDH1A1
SCHEMBL10744129 0.79 AURKA (0.70) AURKAPDE2APRMT5PDE5AFGFR1
SCHEMBL7395290 0.79 AURKA (0.64) AURKAPDE2APDE5AHPSEKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4515796-A INOTROPIC, BRONCHODILATOR, VASODILATORS, ANTICOAGULANTS ELI LILLY AND COMPANY (US) 1985-05-07 US disclosed