SCHEMBL10985132

SCHEMBL10985132

COc1ccc(CCN(C)CCCN2C=Cc3cc(OC)c(OC)cc3CC2=O)cc1OC

nearest known ligand 0.73

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 6/20 0.73
MAPT P10636 1/20 0.63
CYP3A4 P08684 2/20 0.62
ALOX15 P16050 1/20 0.62
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
SMPD1 P17405 5/20 0.52
ABCB1 P08183 1/20 0.52
BLM P54132 1/20 0.51
PMP22 Q01453 1/20 0.51
BRD4 O60885 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10986664 0.99 HCN4 (0.72) HCN4MAPTCYP3A4ALOX15CYP1A2
SCHEMBL11263213 0.97 HCN4 (0.72) HCN4MAPTCYP3A4ALOX15CYP1A2
SCHEMBL10599539 0.94 HCN4 (0.65) HCN4MAPTCYP3A4ALOX15CYP1A2
SCHEMBL10979298 0.94 HCN4 (0.75) HCN4MAPTCYP3A4ALOX15CYP1A2
SCHEMBL11095646 0.93 HCN4 (0.64) HCN4MAPTCYP3A4ALOX15CYP1A2
Hydrochloric Acid SCHEMBL10599369 0.93 HCN4 (0.64) HCN4MAPTCYP3A4ALOX15CYP1A2
Hydrochloric Acid SCHEMBL10983829 0.92 HCN4 (0.63) HCN4MAPTCYP3A4ALOX15CYP1A2
SCHEMBL11092035 0.91 HCN4 (0.61) HCN4MAPTCYP3A4ALOX15SMPD1
Hydrochloric Acid SCHEMBL10984472 0.90 HCN4 (0.60) HCN4MAPTCYP3A4ALOX15SMPD1
SCHEMBL11087721 0.90 HCN4 (0.60) HCN4MAPTCYP3A4ALOX15CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0065229-B1 BENZAZEPINES, PROCESS FOR THEIR PREPARATION AND THEIR APPLICATION AS PHARMACEUTICAL PREPARATIONS Dr. Karl Thomae GmbH (DE) 1985-08-07 EP disclosed
US-4490369-A HYPOTENSIVE, BRRADYCARDIAL DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1984-12-25 US disclosed
EP-0065229-A1 Benzazepines, process for their preparation and their application as pharmaceutical preparations Dr. Karl Thomae GmbH (DE) 1982-11-24 EP disclosed