SCHEMBL11092035

SCHEMBL11092035

COc1ccc(CCN(C)CCCN2C=Cc3cc(OC)c(OC)cc3CC2=O)cc1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 6/20 0.61
MAPT P10636 1/20 0.52
CYP3A4 P08684 1/20 0.52
ALOX15 P16050 1/20 0.52
BRD4 O60885 1/20 0.49
SMPD1 P17405 7/20 0.47
SIGMAR1 Q99720 1/20 0.44
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
ABCB1 P08183 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10984472 0.99 HCN4 (0.60) HCN4MAPTCYP3A4ALOX15BRD4
SCHEMBL10985132 0.91 HCN4 (0.73) HCN4MAPTCYP3A4ALOX15BRD4
Hydrochloric Acid SCHEMBL10986664 0.90 HCN4 (0.72) HCN4MAPTCYP3A4ALOX15BRD4
SCHEMBL11263213 0.88 HCN4 (0.72) HCN4MAPTCYP3A4ALOX15BRD4
SCHEMBL11091288 0.86 HCN4 (0.55) HCN4MAPTCYP3A4ALOX15BRD4
SCHEMBL10599539 0.85 HCN4 (0.65) HCN4MAPTCYP3A4ALOX15BRD4
SCHEMBL10980734 0.85 HCN4 (0.58) HCN4MAPTCYP3A4ALOX15BRD4
SCHEMBL10979298 0.85 HCN4 (0.75) HCN4MAPTCYP3A4ALOX15BRD4
SCHEMBL10977976 0.85 HCN4 (0.54) HCN4MAPTCYP3A4ALOX15BRD4
Hydrochloric Acid SCHEMBL10599369 0.85 HCN4 (0.64) HCN4MAPTCYP3A4ALOX15BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4490369-A HYPOTENSIVE, BRRADYCARDIAL DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1984-12-25 US disclosed
EP-0065229-A1 Benzazepines, process for their preparation and their application as pharmaceutical preparations Dr. Karl Thomae GmbH (DE) 1982-11-24 EP disclosed