SCHEMBL10985990

SCHEMBL10985990

N=C(N)Nc1csc(CO)n1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 10/20 0.36
CDK5R1 Q15078 10/20 0.36
CCNA2 P20248 6/20 0.34
CDK2 P24941 6/20 0.34
CCNA1 P78396 6/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797578 0.78 CDK5 (0.37) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL8796670 0.77 HDAC1 (0.40) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL20557462 0.76 CDK5 (0.43) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL6741408 0.70 CDK5 (0.35) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL22031127 0.68 CDK5 (0.44) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL7332982 0.68 CDK5 (0.58) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL10702053 0.68 SMN1; SMN2 (0.42)
Hydrochloric Acid SCHEMBL10703604 0.67 SMN1; SMN2 (0.41)
SCHEMBL8686075 0.67 CDK5 (0.38) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL6233700 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4492794-A 2-Guanidino-4-hydroxymethylthiazole and derivatives thereof SHIONOGI & CO., LTD. (JP) 1985-01-08 US disclosed
EP-0123741-A1 2-Guanidino-4-hydroxymethylthiazole and derivatives thereof SHIONOGI & CO., LTD. (JP) 1984-11-07 EP disclosed