SCHEMBL6741408

SCHEMBL6741408

N=C(N)Nc1csc(C(=O)O)n1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 4/20 0.35
CDK5R1 Q15078 4/20 0.35
CCNA2 P20248 2/20 0.35
CDK2 P24941 2/20 0.35
CCNA1 P78396 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
NR1H4 Q96RI1 1/20 0.30
GRM5 P41594 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26678642 0.71 PI4KB (0.38) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL10985990 0.70 CDK5 (0.36) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL8797578 0.70 CDK5 (0.37) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL7332982 0.70 CDK5 (0.58) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL8796670 0.69 HDAC1 (0.40) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL6881657 0.69 L3MBTL1 (0.65) L3MBTL1
SCHEMBL5171437 0.69 HCAR3 (0.46) CDK5CDK5R1CA1CA2CA9
SCHEMBL12169124 0.68 HTR2B (0.50) L3MBTL1
Water SCHEMBL7146996 0.68 L3MBTL1 (0.63) L3MBTL1
Hydrochloric Acid SCHEMBL6736638 0.68 L3MBTL1 (0.63) L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040127477-A1 Heterocyclic glycyl beta-alanine derivatives G. D. SEARLE & CO. (US) 2004-07-01 US disclosed
US-6689754-B1 PIPERIDINE OR PYRIDINE DERIVATIVES; ALPHA V BETA 3 INTEGRIN ANTAGONISTS G. D. SEARLE & CO. 2004-02-10 US disclosed
EP-1070060-A1 HETEROCYCLIC GLYCYL BETA-ALANINE DERIVATIVES AS VITRONECTIN ANTAGONISTS G.D. Searle & Co. (US) 2001-01-24 EP disclosed
WO-1999052896-A1 HETEROCYCLIC GLYCYL BETA-ALANINE DERIVATIVES AS VITRONECTIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-10-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040127477-A1 Heterocyclic glycyl beta-alanine derivatives ITGB3, ITGAL, ITGB1 CDK5 2995/4885CDK5R1 2029/4885CCNA2 3811/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.