SCHEMBL10988752

SCHEMBL10988752

CNCCC(Oc1ccc(OC)cc1)C1CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 9/20 0.41
SLC6A2 P23975 4/20 0.41
KDM4E B2RXH2 2/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
GAA P10253 2/20 0.37
MAPK1 P28482 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MAPT P10636 1/20 0.37
CYP2D6 P10635 4/20 0.36
NOS2 P35228 1/20 0.36
CYP2C19 P33261 3/20 0.36
MEN1 O00255 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
TSHR P16473 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 2/20 0.36
SLC6A3 Q01959 2/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10991902 0.88 SLC6A4 (0.40) SLC6A4SLC6A2KDM4EMAPK1MAPT
SCHEMBL10992307 0.86 SLC6A4 (0.54) SLC6A4SLC6A2KDM4EMAPK1CYP2D6
SCHEMBL10985391 0.86 SLC6A4 (0.54) SLC6A4SLC6A2KDM4EMAPK1CYP2D6
SCHEMBL10987185 0.86 SLC6A4 (0.39) SLC6A4SLC6A2KDM4EMAPK1CYP2D6
SCHEMBL10997868 0.86 SLC6A4 (0.54) SLC6A4SLC6A2NOS2SLC6A3SIGMAR1
SCHEMBL10991359 0.86 SLC6A4 (0.39) SLC6A4SLC6A2KDM4EMAPK1CYP2D6
SCHEMBL10993181 0.86 SLC6A4 (0.55) SLC6A4SLC6A2KDM4EMAPK1CYP2D6
SCHEMBL10995043 0.85 MTNR1A (0.48) SLC6A4SLC6A2KDM4EMTNR1AMTNR1B
SCHEMBL10993674 0.84 POLB (0.43) SLC6A4SLC6A2NPSR1MAPTCYP2D6
SCHEMBL10992162 0.84 SLC6A4 (0.39) SLC6A4SLC6A2KDM4EGAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4500541-A Pharmacologically active cyclopropane derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1985-02-19 US disclosed
EP-0039771-B1 CYCLOPROPANE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PRODUCTION MERCK PATENT GmbH (DE) 1983-10-19 EP disclosed