SCHEMBL10991925

SCHEMBL10991925

CCCc1c(F)c(F)c(C(=O)O)c(F)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 3/20 0.42
LDHB P07195 3/20 0.42
HCAR2 Q8TDS4 3/20 0.40
PTPN1 P18031 1/20 0.39
PTPN11 Q06124 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.37
PKM P14618 1/20 0.37
ESR1 P03372 1/20 0.34
JUN P05412 1/20 0.34
METAP2 P50579 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
BID P55957 3/20 0.32
MCL1 Q07820 3/20 0.32
BCL2L1 Q07817 2/20 0.32
BAK1 Q16611 2/20 0.32
KAT8 Q9H7Z6 2/20 0.32
PPARG P37231 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7855502 0.89 LDHA (0.41) LDHALDHBHCAR2PTPN1PTPN11
SCHEMBL10981379 0.82 SMN1; SMN2 (0.39) LDHALDHBHCAR2SMN1; SMN2PKM
SCHEMBL5586968 0.80 LDHA (0.49) LDHALDHBHCAR2PTPN1PTPN11
Alcohol SCHEMBL29191762 0.79 SMN1; SMN2 (0.43) HCAR2PTPN1PTPN11SMN1; SMN2PKM
SCHEMBL22418967 0.79 LDHA (0.48) LDHALDHBHCAR2PTPN1PTPN11
SCHEMBL14989236 0.79 LDHA (0.48) LDHALDHBHCAR2PTPN1PTPN11
SCHEMBL11936748 0.78 SMN1; SMN2 (0.41) HCAR2SMN1; SMN2PKMESR1MEN1
SCHEMBL27417437 0.78 TAAR1 (0.39)
SCHEMBL29927198 0.78 HCAR2 (0.47) LDHALDHBHCAR2SMN1; SMN2PKM
SCHEMBL7855513 0.78 HCAR2 (0.47) LDHALDHBHCAR2SMN1; SMN2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4551546-A INSECTICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-11-05 US disclosed
US-4429153-A INSECTICIDES, MITICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-01-31 US disclosed
EP-0031199-B1 SUBSTITUTED BENZYL ESTERS OF CYCLOPROPANE CARBOXYLIC ACIDS AND THEIR PREPARATION, COMPOSITIONS CONTAINING THEM AND METHODS OF COMBATING INSECT PESTS THEREWITH, AND SUBSTITUTED BENZYL ALCOHOLS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-12-14 EP disclosed
US-4405640-A Substituted fluorobenzyl cyclopropane carboxylates useful as insecticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-09-20 US disclosed
EP-0060617-A1 Fluorobenzyl cyclopropane carboxylates, their preparation, compositions and use as insecticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-09-22 EP disclosed
EP-0031199-A1 Substituted benzyl esters of cyclopropane carboxylic acids and their preparation, compositions containing them and methods of combating insect pests therewith, and substituted benzyl alcohols IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1981-07-01 EP disclosed