SCHEMBL11004271

SCHEMBL11004271

Cc1cncc(-c2c[nH]c(=O)c(N)c2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 10/20 0.54
INCENP Q9NQS7 10/20 0.54
TTK P33981 9/20 0.54
AURKA O14965 8/20 0.54
MAPT P10636 2/20 0.50
THRB P10828 2/20 0.50
CASP1 P29466 2/20 0.50
PDE3B Q13370 2/20 0.50
PDE3A Q14432 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50
CYP1A2 P05177 1/20 0.50
GLA P06280 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
HPGD P15428 1/20 0.50
ALOX15 P16050 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10998739 0.84 TTK (0.57) AURKBINCENPTTKAURKAMAPT
SCHEMBL11000281 0.82 TTK (0.54) AURKBINCENPTTKAURKAMAPT
SCHEMBL10996933 0.81 TTK (0.55) AURKBINCENPTTKAURKAMAPT
SCHEMBL11003225 0.81 TTK (0.50) AURKBINCENPTTKAURKAMAPT
SCHEMBL11002890 0.80 CYP11B1 (0.36) AURKBINCENPTTKAURKACYP11B1
SCHEMBL11448065 0.80 AURKB (0.50) AURKBINCENPTTKAURKAMAPT
SCHEMBL11000547 0.78 CYP11B2 (0.56) PDE3BPDE3AKDM4EALDH1A1LMNA
SCHEMBL10995582 0.78 AURKB (0.51) AURKBINCENPTTKAURKAMAPT
SCHEMBL11458612 0.76 AURKB (0.57) AURKBINCENPTTKAURKAMAPT
SCHEMBL11001428 0.75 TTK (0.59) AURKBINCENPTTKAURKAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4514400-A Cardiotonic 5-heteroaryl-pyridone WILLIAM H. RORER, INC. (US) 1985-04-30 US disclosed